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  • Alessia Distefano, Paolo Corsaro, Nunzio Tuccitto, Francesca Laneri, Olivier Monasson, et al.. Intrinsically photoluminescent hydrogels to measure peptides‑copper binding affinities. Journal of Inorganic Biochemistry, 2025, 268, pp.112914. ⟨10.1016/j.jinorgbio.2025.112914⟩. ⟨hal-05052019⟩
  • Mayssa Zayene, Franck Le Bideau, Pascal Retailleau, Hichem Ben Jannet, Vincent Gandon, et al.. Dual Photoredox/Cu‐Catalysis Enables Diastereoselective Synthesis of 3‐ β ‐Ethynyltropanes via Decarboxylative Alkynylation. Advanced Synthesis and Catalysis, 2025, ⟨10.1002/adsc.202500241⟩. ⟨hal-05114385⟩
  • Ömer Taspinar, Daniel J Leonard, Nathan Picois, Cornelia Göcke, Matej Žabka, et al.. Asymmetric Intramolecular α‐Arylation of Polar Amino Acids Bearing β‐Leaving Groups. Angewandte Chemie International Edition, 2025, ⟨10.1002/anie.202507713⟩. ⟨hal-05110334⟩
  • Monika Skibinska, Alicja Warowicka, Benoît Crousse, Tomasz Cytlak. Synthesis and Antibacterial Activity of Novel Phosphonated CF 3 -β-lactams. ACS Omega, 2025, 10 (17), pp.18062-18072. ⟨10.1021/acsomega.5c01562⟩. ⟨hal-05105385⟩
  • Sarah Szwarc, Adriano Rutz, Kyungha Lee, Yassine Mejri, Olivier Bonnet, et al.. Translating community-wide spectral library into actionable chemical knowledge: a proof of concept with monoterpene indole alkaloids. Journal of Cheminformatics, 2025, 17, pp.62. ⟨10.1186/s13321-025-01009-0⟩. ⟨hal-05058394⟩
  • Xinya Liu, Valentin Dorokhov, Olivier Provot, Christine Tran, Pascal Retailleau, et al.. Mechanochemical Approach for Metal‐Free Regioselective C5‐Sulfenylation of Imidazo[2,1‐b]thiazoles. ChemSusChem, 2025, ⟨10.1002/cssc.202500320⟩. ⟨hal-05053681⟩
  • Jun Yan, Pascal Retailleau, Abdallah Hamze, Christine Tran. Copper‐Catalyzed Domino Synthesis of Spiropyrazoline Oxindoles via Condensation of Indolin‐2‐One and Phenylhydrazine Derivatives. Advanced Synthesis and Catalysis, 2025, 367 (10), ⟨10.1002/adsc.202500223⟩. ⟨hal-05127035⟩
  • Davide Di Lorenzo, Nicolo Bisi, Raffaella Bucci, Inga Ennen, Leonardo Lo Presti, et al.. Application of modular isoxazoline-β$^{2,2-}$amino acid-based peptidomimetics as chemical model systems for studying the tau misfolding. iScience, 2025, 28 (4), pp.112272. ⟨10.1016/j.isci.2025.112272⟩. ⟨hal-05056022⟩
  • Florent Edde, Emmanuelle Drège, Laurent Evanno. User‐friendly and Green Procedure for a Photoinduced Wohl‐Ziegler Reaction. European Journal of Organic Chemistry, 2025, 28 (18), ⟨10.1002/ejoc.202500183⟩. ⟨hal-05114321⟩
  • Mathew Choaji, Ascel Samba-Louaka, Zineb Fechtali-Moute, Willy Aucher, Sébastien Pomel. Encystment and Excystment Processes in Acanthamoeba castellanii: An Emphasis on Cellulose Involvement. Pathogens, 2025, 14, ⟨10.3390/pathogens14030268⟩. ⟨hal-04988818⟩
  • Shashank Pandey, Elisa Peroni, Dagmar Jarkovska, Magdalena Chottova Dvorakova, Olivier Monasson, et al.. Role of Neuropeptide B/W Signaling in Modulating Intracellular Calcium in Human Skin Fibroblasts. Frontiers in Bioscience-Landmark, 2025, 30 (2), ⟨10.31083/FBL26760⟩. ⟨hal-04971764⟩
  • Alicia Maroto, Olivier Briand, Alessia Distefano, Filiz Arioz, Olivier Monasson, et al.. Differentiation of Isomeric TAT1-CARNOSINE Peptides by Energy-Resolved Mass Spectrometry and Principal Component Analysis. Molecules, 2025, Special Issue Design, Synthesis, and Analysis of Potential Drugs, 3rd Edition, 30 (4), pp.853. ⟨10.3390/molecules30040853⟩. ⟨hal-04943837⟩
  • Marion Alter, Margherita Donnici, Solenn Reguer, Mathieu Thoury, Matthieu Réfrégiers, et al.. Alteration markers of green copper bimetallic pigments in easel paintings by an inter-comparison of analogues and historical samples. Microchemical Journal, 2025, 209, pp.112541. ⟨10.1016/j.microc.2024.112541⟩. ⟨hal-04942544⟩
  • Louis-Valentin Méteignier, Sarah Szwarc, Patra Barunava, Mickael Durand, Duchesse-Lacours Zamar, et al.. Harnessing the spatial and transcriptional regulation of monoterpenoid indole alkaloid metabolism in Alstonia scholaris leads to the identification of broad geissoschizine cyclase activities. Plant Physiology and Biochemistry, 2025, 219, pp.109363. ⟨10.1016/j.plaphy.2024.109363⟩. ⟨hal-04810555⟩
  • Bastien Champciaux, Nicolas Jamey, Bruno Figadère, Laurent Ferrié. Peroxycarbenium-Mediated Asymmetric Synthesis of 1,2-Dioxanes and 1,2-Dioxolanes. Journal of the American Chemical Society, 2025, 147 (4), pp.3353-3359. ⟨10.1021/jacs.4c13899⟩. ⟨hal-04918894⟩
  • Marceau Levasseur, Alice Trac, Isabelle Clavereau, Flavien Zannini, Yannick Estevez, et al.. Reverse chemical ecology to study the defense of the plant host Sextonia rubra and the chemical mediators of its endophyte Fusarium falciforme against phytopathogen Trametes versicolor. Phytochemistry, 2025, 238, pp.114577. ⟨10.1016/j.phytochem.2025.114577⟩. ⟨hal-05128635⟩
  • Lorenzo Meneghelli, Stephanie Davidson, Anthony Gineste, Lamia El Guermah, Sabrina Kellouche-Gaillard, et al.. Design and synthesis of a clickable cell-permeable pseudopeptide Pin1 inhibitor with antiproliferative effects on human multiple myeloma cell line. Chemical Communications, 2025, ⟨10.1039/D4CC05968A⟩. ⟨hal-05003977⟩
  • Yuqing Zhang, Myriam Eveno, Nadège Lubin-Germain, Agnès Lattuati-Derieux, Nadège Lubin-Germain, et al.. Partially fluorinated derivatives as a powerful tool for the restoration of blanched easel paintings. Progress in Organic Coatings, 2025, 207, pp.109375. ⟨10.1016/j.porgcoat.2025.109375⟩. ⟨hal-05104320⟩
  • Rany B. Mbeng Obame, Sidney Gallard, Sacha Gibert, Jean-François Gallard, Solenn Ferron, et al.. Unifying the Absolute Configuration of Dibenzopyrrocoline Alkaloids with Relative Configuration Revision of Cryptowolinol and Description of Isocryptaustoline from Cryptocarya oubatchensis. Journal of Natural Products, 2025, ⟨10.1021/acs.jnatprod.4c01315⟩. ⟨hal-05024657⟩
  • Farzin Arjmand, Alima Chali, Youssef Snoussi, David Troadec, Gilles Patriarche, et al.. In-situ chemical grafting of aminophenyl and RGD peptide on an equimolar high-entropy HfNbTaTiZr alloy: electrochemical behavior and surface characterization. Emergent Materials, 2024, ⟨10.1007/s42247-024-00963-z⟩. ⟨hal-04854358⟩
  • Norbert Hoffmann, Mario Andrés Gomez Fernandez, Arthur Desvals, Corentin Lefebvre, Clément Michelin, et al.. Photochemical reactions of biomass derived platform chemicals. Frontiers in Chemistry, 2024, 12, ⟨10.3389/fchem.2024.1485354⟩. ⟨hal-04831095⟩
  • Julien Pytkowicz, Grégory Chaume, Nathalie Lensen, Evelyne Chelain, Thierry Brigaud. Two decades of fluorine chemistry in Cergy. Comptes Rendus. Chimie, 2024, 27 (G1), pp.353-383. ⟨10.5802/crchim.360⟩. ⟨hal-04823676⟩
  • Sarah Szwarc, Pierre Le Pogam, Mehdi Beniddir. Emerging trends in plant natural products biosynthesis: a chemical perspective. Current Opinion in Plant Biology, 2024, 82, pp.102649. ⟨10.1016/j.pbi.2024.102649⟩. ⟨hal-05058399⟩
  • Enzo Lezin, Mickael Durand, Caroline Birer Williams, Ana Luisa Lopez Vazquez, Thomas Perrot, et al.. Genome‐based discovery of pachysiphine synthases in Tabernaemontana elegans. The Plant Journal, 2024, 120 (5), pp.1880-1900. ⟨10.1111/tpj.17085⟩. ⟨hal-05036872⟩
  • Gulsah Bayraktar, Pascal Marchand, Euzébio Guimarães Barbosa, Marilia Cecilia da Silva, Karen Cacilda Weber, et al.. Biological properties and in silico studies of thiazolopyrimidine derivatives active against visceral and cutaneous Leishmania spp. amastigote forms. European Journal of Medicinal Chemistry Reports, 2024, 12, pp.100228. ⟨10.1016/j.ejmcr.2024.100228⟩. ⟨hal-05088062⟩
  • Aurélie Honfroy, Jolien Bertouille, Ana-Maria Turea, Thibault Cauwenbergh, Jessica Bridoux, et al.. Fluorinated Peptide Hydrogels Result in Longer In Vivo Residence Time after Subcutaneous Administration. Biomacromolecules, 2024, 25 (10), pp.6666-6680. ⟨10.1021/acs.biomac.4c00872⟩. ⟨hal-04782661⟩
  • Nalia Mekarnia, Kamal-Eddine Benallal, Jovana Sádlová, Barbora Vojtková, Aurélie Mauras, et al.. Effect of Phlebotomus papatasi on the fitness, infectivity and antimony-resistance phenotype of antimony-resistant Leishmania major Mon-25. International journal for parasitology. Drugs and drug resistance, 2024, 25, pp.100554. ⟨10.1016/j.ijpddr.2024.100554⟩. ⟨hal-04632483⟩
  • Pieter Langerhorst, Melissa Baerenfaenger, Purva Kulkarni, Simon Nadal, Charissa Wijnands, et al.. N-linked glycosylation of the M-protein variable region: glycoproteogenomics reveals a new layer of personalized complexity in multiple myeloma. Clinical Chemistry and Laboratory Medicine, 2024, 62 (8), pp.1626-1635. ⟨10.1515/cclm-2023-1189⟩. ⟨hal-05085563⟩
  • Dimitra Kyrko, Murat Saraç, Jing Hao, Pascal Retailleau, Sandrine Ongeri, et al.. Functionalized α‐Fluorinated Amines from Imines and Enol Ethers. Advanced Synthesis and Catalysis, 2024, 366 (16), pp.3460-3465. ⟨10.1002/adsc.202400517⟩. ⟨hal-04756974⟩
  • Farzin Arjmand, Adrien Mourgout, Alima Chali, Madjid Djemai, Credson-Yannick Langueh, et al.. L-PBF processing and characterization of a Ti 35 Nb 30 Zr 29 Mo 3 Ta 3 multiprincipal element alloy for medical implants. Applied Physics Letters, 2024, 125 (4), pp.041904. ⟨10.1063/5.0208341⟩. ⟨hal-04739764⟩
  • Yu Fan, Ahmed El Rhaz, Stéphane Maisonneuve, Emilie Gillon, Maha Fatthalla, et al.. Photoswitchable glycoligands targeting Pseudomonas aeruginosa LecA. Beilstein Journal of Organic Chemistry, 2024, 20, pp.1486-1496. ⟨10.3762/bjoc.20.132⟩. ⟨hal-04637573⟩
  • Nicolas Jamey, Laurent Ferrié. Stereodivergent Total Synthesis of Ethyl Plakortide Z. Organic Letters, 2024, 26 (27), pp.5741-5745. ⟨10.1021/acs.orglett.4c01893⟩. ⟨hal-04738657⟩
  • Clémence Rose, Rodrigo Hernán Tomas‐grau, Brenda Zabala, Patrick Pierre Michel, Jean‐michel Brunel, et al.. C9‐Functionalized Doxycycline Analogs as Drug Candidates to Prevent Pathological α‐Synuclein Aggregation and Neuroinflammation in Parkinson's Disease Degeneration. ChemMedChem, 2024, 19, ⟨10.1002/cmdc.202300597⟩. ⟨hal-04736533⟩
  • Ivanna Amarsy, Nicolas Gigant, Izel D Erturk, Nicolas Bogliotti, Delphine Joseph, et al.. Palladium‐Catalyzed Indirect and Regioselective Phosphonation of Azobenzenes: Toward the Design of Water‐Soluble Photoswitches. European Journal of Organic Chemistry, 2024, 27 (28), pp.e202400406. ⟨10.1002/ejoc.202400406⟩. ⟨hal-04739274⟩
  • Diana Lamaa, Catherine Cailleau, Juliette Vergnaud, Julie Mougin, Jérôme Bignon, et al.. Overcoming Solubility Challenges: Liposomal isoCoQ‐Carbazole as a Promising Anti‐Tumor Agent for Inoperable and Radiation‐Insensitive cancers. ChemBioChem, 2024, ⟨10.1002/cbic.202400062⟩. ⟨hal-04569859⟩
  • Benoit Derrien, Karine Leblanc, Laurent Evanno, Emmanuelle Drège. Enantioselective Total Synthesis of the Neurotoxin Caramboxin. Journal of Organic Chemistry, 2024, 89 (9), pp.6489-6493. ⟨10.1021/acs.joc.4c00541⟩. ⟨hal-05114333⟩
  • Zuzana Palčeková, Kavita De, Shiva Kumar Angala, Martine Gilleron, Sophie Zuberogoïtia, et al.. Impact of methylthioxylose substituents on the biological activities of lipomannan and lipoarabinomannan in Mycobacterium tuberculosis. ACS Infectious Diseases, 2024, 10 (4), pp.1379-1390. ⟨10.1021/acsinfecdis.4c00079⟩. ⟨hal-04725853⟩
  • Chloé Breton-Patient, Sébastien Billotte, Patricia Duchambon, Gaëlle Fontaine, Sophie Bombard, et al.. Light‐Activatable Photocaged UNC2025 for Triggering TAM Kinase Inhibition in Bladder Cancer. ChemBioChem, 2024, 25 (8), pp.e202300855. ⟨10.1002/cbic.202300855⟩. ⟨hal-04783958⟩
  • Luca Paoletti, Francesco Baschieri, Claudia Migliorini, Chiara Di Meo, Olivier Monasson, et al.. 3D printing of gellan‐dextran methacrylate IPNs in glycerol and their bioadhesion by RGD derivatives. Journal of Biomedical Materials Research Part A, 2024, ⟨10.1002/jbm.a.37698⟩. ⟨hal-04488395⟩
  • Eric Konofal, Michel Lecendreux, Jean-Charles Bizot, Anh-Tuan Lormier, Bruno Figadère. NLS-3 (Levophacetoperane or (R,R) Phacetoperane): A Reverse Ester of Methylphenidate: A Literature Review. Current Medicinal Chemistry, 2024, 31 (9), pp.1069-1081. ⟨10.2174/0929867330666230120161837⟩. ⟨hal-04284826⟩
  • Muhammad Tahir Muhammad, Mehdi Beniddir, Lacksany Phongphane, Mohamad Hafizi Abu Bakar, Mohd Hazwan Hussin, et al.. Chemodiverse monoterpene indole alkaloids from Kopsia teoi, inhibitory potential against α-amylase, and their molecular docking studies. Fitoterapia, 2024, 174, pp.105873. ⟨10.1016/j.fitote.2024.105873⟩. ⟨hal-04490024⟩
  • Nicolò Bisi, Luca Pinzi, Giulio Rastelli, Nicolo Tonali. Early Diagnosis of Neurodegenerative Diseases: What Has Been Undertaken to Promote the Transition from PET to Fluorescence Tracers. Molecules, 2024, 29 (3), pp.722. ⟨10.3390/molecules29030722⟩. ⟨hal-04523467⟩
  • Francesco Terzani, Sherazade Belhattab, Aurore Le Guern, Karine Guitot, Olivier Monasson, et al.. Synthesis and biological evaluation of selective Pepstatin based trifluoromethylated inhibitors of Cathepsin D. European Journal of Medicinal Chemistry, 2024, 267, pp.116178. ⟨10.1016/j.ejmech.2024.116178⟩. ⟨hal-04455850⟩
  • Monika Skibinska, Alicja Warowicka, Henryk Koroniak, Tomasz Cytlak, Benoît Crousse. Synthesis, Reactivity, and Antibacterial Activity of gem -Difluoroalkene, Difluoromethyl, and Trifluoromethyl β-Lactams. Organic Letters, 2024, 26 (3), pp.692-696. ⟨10.1021/acs.orglett.3c04094⟩. ⟨hal-04756963⟩
  • Ning Liu, Ping Gao, Hai-Yan Lu, Lei Fang, Julien Nicolas, et al.. Polyfluoroalkyl Chain‐Based Assemblies for Biomimetic Catalysis. Chemistry - A European Journal, In press, 30 (1), ⟨10.1002/chem.202302669⟩. ⟨hal-04252759⟩
  • Wafa Redjdal, Sara Benmahdjoub, Thi Thanh Hyen Luong, Belkacem Benmerad, Franck Le Bideau, et al.. Pd‐Catalyzed Coupling of Bromo‐N‐(β‐glucopyranosyl)quinolin‐2‐ones with Amides: Synthesis of N‐glucosyl‐6BrCaQ Conjugates with Potent Anticancer Activity. ChemMedChem, 2024, 19 (15), pp.e202400195. ⟨10.1002/cmdc.202400195⟩. ⟨hal-04905231⟩
  • Nathan Picois, Yazid Boutahri, Pierre Milbeo, Chiara Zanato, Nathalie Lensen, et al.. Asymmetric α-Fluoroalkyl-α-Amino Acids: Recent Advances in Their Synthesis and Applications. Molecules, 2024, 29 (6), pp.1408. ⟨10.3390/molecules29061408⟩. ⟨hal-04516441⟩
  • Ismaila Ciss, Matar M Seck, Bruno Figadère, Laurent Ferrié. Advances Toward Amphidinolides C, F and U: Isolations, Synthetic Studies and Total Syntheses. Chemistry - A European Journal, 2024, 30 (27), pp.e202400471. ⟨10.1002/chem.202400471⟩. ⟨hal-04738667⟩
  • José Laxio Arenas, Jacopo Lesma, Tap Ha‐duong, Bikash Ranjan Sahoo, Ayyalusamy Ramamoorthy, et al.. Composition and Conformation of Hetero‐ versus Homo‐Fluorinated Triazolamers Influence their Activity on Islet Amyloid Polypeptide Aggregation. Chemistry - A European Journal, 2024, 30 (28), pp.e202303887. ⟨10.1002/chem.202303887⟩. ⟨hal-04756674⟩
  • Linhua Shen, Franck Le Bideau, Gong Chen, Samir Messaoudi. Pd-catalyzed S -glycosylation of cysteine-containing peptides at room temperature. Organic Chemistry Frontiers, 2024, 11 (22), pp.6347-6352. ⟨10.1039/d4qo01389a⟩. ⟨hal-04905247⟩
  • Imen Abid, Wassim Moslah, Sandrine Cojean, Nicolas Imbert, Philippe M Loiseau, et al.. The Synthesis of 2′-Hydroxychalcones under Ball Mill Conditions and Their Biological Activities. Molecules, 2024, 29 (8), pp.1819. ⟨10.3390/molecules29081819⟩. ⟨hal-04550832⟩
  • Olivier Provot. Novel access to α-carbolines with biological applications. European Journal of Medicinal Chemistry, 2024, 276, pp.116700. ⟨10.1016/j.ejmech.2024.116700⟩. ⟨hal-04697354⟩
  • Nathan Picois, Lizeth Bodero, Pierre T Milbeo, Thierry Brigaud, Grégory Chaume. Bimodal use of chiral α‐Trifluoromethylalanine in Aib Foldamers: study of the position impact towards the helical screw‐sense preference. Chemistry - A European Journal, In press, ⟨10.1002/chem.202400540⟩. ⟨hal-04516499⟩
  • Gaël Printz, Redoy Gazi Shuvo, Antoine Schweizer, Dmytro Ryzhakov, Christophe Gourlaouen, et al.. N-Heterocyclic carbene-initiated epoxide/anhydride ring-opening copolymerization: effective and selective organoinitiators for the production of various polyesters. Polymer Chemistry, 2024, 15 (38), pp.3901 - 3906. ⟨10.1039/d4py00778f⟩. ⟨hal-04896594v2⟩
  • Chloé Cayrou, Astrid Walrant, Delphine Ravault, Karine Guitot, Sylvie Noinville, et al.. Incorporation of CF 3 -pseudoprolines into polyproline type II foldamers confers promising biophysical features. Chemical Communications, In press, ⟨10.1039/D4CC02895C⟩. ⟨hal-04660873⟩
  • Ping Gao, Tâp Ha-Duong, Julien Nicolas. Coarse‐Grained Model‐Assisted Design of Polymer Prodrug Nanoparticles with Enhanced Cytotoxicity: A Combined Theoretical and Experimental Study. Angewandte Chemie, 2024, ⟨10.1002/ange.202316056⟩. ⟨hal-04468750⟩
  • David Meijer, Mehdi A Beniddir, Connor W Coley, Yassine M Mejri, Meltem Öztürk, et al.. Empowering natural product science with AI: leveraging multimodal data and knowledge graphs. Natural Product Reports, In press, ⟨10.1039/d4np00008k⟩. ⟨hal-04700044⟩
  • Thibault Gendron, Don Antoine Lanfranchi, Nicole I Wenzel, Hripsimée Kessedjian, Beate Jannack, et al.. Chemoselective Synthesis and Anti-Kinetoplastidal Properties of 2,6-Diaryl-4H-tetrahydro-thiopyran-4-one S-Oxides: Their Interplay in a Cascade of Redox Reactions from Diarylideneacetones. Molecules, 2024, 29 (7), pp.1620. ⟨10.3390/molecules29071620⟩. ⟨hal-04583951⟩
  • Pierre Le Pogam, Mehdi Beniddir. Structural diversity and chemical logic underlying the assembly of monoterpene indole alkaloids oligomers. Natural Product Reports, 2024, 41 (11), pp.1723-1765. ⟨10.1039/D4NP00011K⟩. ⟨hal-05058404⟩
  • Dongxu Zhai, Shuxin Yan, James Samsom, Le Wang, Ping Su, et al.. Small-molecule targeting AMPA-mediated excitotoxicity has therapeutic effects in mouse models for multiple sclerosis. Science Advances , 2023, 9 (49), ⟨10.1126/sciadv.adj6187⟩. ⟨hal-04604036⟩
  • Linhua Shen, Olivier Monasson, Elisa Peroni, Franck Le Bideau, Samir Messaoudi. Electrochemical Nickel-Catalyzed Selective Inter-and Intramolecular Arylations of Cysteine-Containing Peptides. Angewandte Chemie International Edition, 2023, 62 (50), ⟨10.1002/anie.202315748⟩. ⟨hal-04905239v2⟩
  • Cyrille Kouklovsky, Erwan Poupon, Laurent Evanno, Guillaume Vincent. Total Synthesis of Mavacuran Alkaloids with Bioinspired and non-Bioinspired Strategies. SYNLETT, 2023, ⟨10.1055/s-0042-1751498⟩. ⟨hal-04274139⟩
  • Sameh Obeid, Eloisa Berbel-Manaia, Valérie Nicolas, Indira Dennemont, Julien Barbier, et al.. Deciphering the mechanism of action of VP343, an antileishmanial drug candidate, in Leishmania infantum. iScience, 2023, 26 (11), pp.108144. ⟨10.1016/j.isci.2023.108144⟩. ⟨hal-04304917⟩
  • Gaël Printz, Dmytro Ryzhakov, Christophe Gourlaouen, Béatrice Jacques, Samir Messaoudi, et al.. First Use of Thiosquaramides as Polymerization Catalysts: Controlled ROP of Lactide Implicating Key Secondary Interactions for Optimal Performance. ChemCatChem, In press, ⟨10.1002/cctc.202301207⟩. ⟨hal-04295776⟩
  • Mansour Kerim, Laurent Evanno, Laurent Ferrié. Stereodivergent Total Syntheses of (+)-Mycaperoxides C, D, G Methyl Ester and (-)-Mycaperoxide B. Chemistry - A European Journal, 2023, 29 (6), ⟨10.1002/chem.202203004⟩. ⟨hal-04250595⟩
  • William Godefroy, Lionel Faivre, Caroline Sansac, Briac Thierry, Jean-Marc Allain, et al.. Development and qualification of clinical grade decellularized and cryopreserved human esophagi. Scientific Reports, 2023, 13, pp.18283. ⟨10.1038/s41598-023-45610-5⟩. ⟨hal-04269788⟩
  • Camille Lozada, Simon Gonzalez, Rémy Agniel, Mathilde Hindie, Luca Manciocchi, et al.. Introduction of constrained Trp analogs in RW9 modulates structure and partition in membrane models. Bioorganic Chemistry, 2023, 139, pp.106731. ⟨10.1016/j.bioorg.2023.106731⟩. ⟨hal-04272386⟩
  • Francesca Nuti, Maud Larregola, Agnieszka Staśkiewicz, Bernhard Retzl, Nataša Tomašević, et al.. Design, synthesis, conformational analysis, and biological activity of Cα1-to-Cα6 1,4- and 4,1-disubstituted 1H-[1,2,3]triazol-1-yl-bridged oxytocin analogues. Journal of Enzyme Inhibition and Medicinal Chemistry, 2023, 38 (1), pp.2254019. ⟨10.1080/14756366.2023.2254019⟩. ⟨hal-04605577⟩
  • Zuzana Palčeková, Andrés Obregón-Henao, Kavita De, Amanda Walz, Ha Lam, et al.. Role of succinyl substituents in the mannose-capping of lipoarabinomannan and control of inflammation in Mycobacterium tuberculosis infection. PLoS Pathogens, 2023, 19 (9), pp.e1011636. ⟨10.1371/journal.ppat.1011636⟩. ⟨hal-04238654⟩
  • Siwar Soltani, Imed Koubaa, Sandrine Cojean, Carine Picot, Pascal Marchand, et al.. Phytochemical, antileishmanial, antifungal and cytotoxic profiles of Thymelaea tartonraira (L.) All. extracts. Natural Product Research, 2023, 38 (20), pp.3481-3487. ⟨10.1080/14786419.2023.2252153⟩. ⟨hal-04805245⟩
  • Karen Thompson, Sonia Watson, Chiara Zanato, Sergio Dall'Angelo, Joriene de Nooij, et al.. The atypical ‘hippocampal’ glutamate receptor coupled to phospholipase D that controls stretch‐sensitivity in primary mechanosensory nerve endings is homomeric purely metabotropic GluK2. Experimental Physiology, 2023, ⟨10.1113/EP090761⟩. ⟨hal-04273805⟩
  • Huibin Wang, Sébastien Halary, Charlotte Duval, Cécile Bernard, Marc Troussellier, et al.. Diversity, metabolome profiling and bioactivities of benthic filamentous cyanobacteria isolated from coastal mangroves of Mayotte. Frontiers in Marine Science, 2023, 10, ⟨10.3389/fmars.2023.1201594⟩. ⟨mnhn-04174558⟩
  • A. Breine, K. van Holsbeeck, C. Martin, S. Gonzalez, M. Mannes, et al.. Bypassing the Need for Cell Permeabilization: Nanobody CDR3 Peptide Improves Binding on Living Bacteria. Bioconjugate Chemistry, 2023, 34 (7), pp.1234-1243. ⟨10.1021/acs.bioconjchem.3c00116⟩. ⟨hal-04607026⟩
  • Yuqing Zhang, Myriam Eveno, Florian Gallier, Mara Camaiti, Agnès Lattuati-Derieux, et al.. Synthesis of novel partially perfluorinated C-glycosides and their application in blanching easel painting restoration. Journal of Cultural Heritage, 2023, 62, pp.493-500. ⟨10.1016/j.culher.2023.06.019⟩. ⟨hal-04172828⟩
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  • Antoine Gamet, Ismaila Ciss, Bastien Nay. Total synthesis of photoactivatable latrunculin B for actin-targeting chemical biology. Rencontres de Chimie Organique, Apr 2024, Palaiseau (Université Paris-Saclay), France. ⟨hal-04575270⟩
  • Olivier Monasson, Alima Chali, Sonia Touharia, Adrien Mourgout, Farzin Arjmand, et al.. Novel biocompatible alloys via peptides surface engineering. A decade of Peptide Materials, Oct 2023, Sorrento, Italy. . ⟨hal-04725375⟩
  • David Rondeau, Thomas Delhaye, Erell Froger, Yves Gimbert, Axel Raux, et al.. Proposition of optimization strategies in collision energies on QTOF and Orbitrap instruments to perform comparable CID-MS-MS spectra in metabolomics. 39ème Journées Françaises de Spectrométrie de Masse (SFSM 2023 ), Sep 2023, Marseille, France. 2023. ⟨hal-04328759⟩
  • Enzo Lezin, Sarah Szwarc, Louis-Valentin Méteignier, Duchesse-Lacours Zamar, Caroline Birer Williams, et al.. The CYP71 Geissoschizine Cyclase catalyzes multiple cyclisation reactions in the synthesis of monoterpene indole alkaloids. P450 Biodiversity and Biotechnology, 2023, Copenhagen, Denmark. ⟨hal-05056241⟩
  • Sokaina Hammoud, Carine Maaliki, Bastien Champciaux, Albertus Viljoen, Clement Raynaud, et al.. Synthesis and evaluation of heterocycle structures as potential inhibitors of Mycobacterium tuberculosis. Journées de Chimie Organique, Nov 2022, Palaiseau (Ecole Polytechnique), France. ⟨hal-05019003⟩
  • Enzo Lezin, Louis-Valentin Méteignier, Caroline Birer-Williams, Christelle Dutilleul, Arnaud Lanoue, et al.. Elucidating missing steps in the synthesis of the nootropic alkaloid vincamine and production of vincamine-derivatives by human P450s. 34eme colloque BioTechnoCentre, 2022, Nouan-le-Fuzelier, France. ⟨hal-05056191⟩
  • Louis-Valentin Méteignier, Caroline Birer Williams, Mehdi A. Beniddir, Pierre Le Pogam, Christelle Dutilleul, et al.. Transcriptomics in a tropical tree identify a P450 catalyzing distinct cyclizations of monoterpene indole alkaloids. 33eme colloque BioTechnoCentre, 2021, Chaumont sur Tharonne, France. ⟨hal-05055979⟩

Proceedings/Recueil des communications1 document

  • Lorenzo Meneghelli, Lamia El Guermah, Maud Larregola, Sabrina Kellouche-Gaillard, Franck Carreiras, et al.. Design and Synthesis of Pin1-PROTACs as Potential Therapeutic Tools for Cancer Treatment. 36th European Peptide Symposium, Aug 2022, Sitges (Barcelona), Spain. The European Peptide Society, pp.285-287, 2022, ⟨10.17952/36EPS/36EPS.2022.285⟩. ⟨hal-05003974⟩

Chapitres d'ouvrage8 document

  • Thierry Brigaud, B. Crousse, T. Lequeux. Perfluoroalkylated Biomolecules for Medicinal Chemistry and Biological Studies. Perfluoroalkyl Substances, The Royal Society of Chemistry; The Royal Society of Chemistry, pp.459-476, 2022, ⟨10.1039/9781839167591-00459⟩. ⟨hal-04098116⟩
  • Pierre Le Pogam, Erwan Poupon, Pierre Champy, Mehdi Beniddir. Implementation of an MS/MS Spectral Library for Monoterpene Indole Alkaloids. Catharanthus roseus, 2505, Springer US, pp.87-100, 2022, Methods in Molecular Biology, ⟨10.1007/978-1-0716-2349-7_7⟩. ⟨hal-05058417⟩
  • Angélique Ferry, Xavier Guinchard. Bicyclic 5-5 Systems With One Bridgehead (Ring Junction) Nitrogen Atom: Two Extra Heteroatoms 1:1. Comprehensive Heterocyclic Chemistry IV, Elsevier, pp.95-144, 2022, ⟨10.1016/B978-0-12-409547-2.14934-0⟩. ⟨hal-04102152⟩
  • Laurent Ferrié. Advances in the synthesis of 1,2-dioxolanes and 1,2-dioxanes. Eric F.V. Scriven; Christopher A. Ramsden. Advances in Heterocyclic Chemistry, 135, Elsevier, pp.57-146, 2021, 978-0-12-824619-1. ⟨10.1016/bs.aihch.2021.03.001⟩. ⟨hal-03320615⟩
  • Angélique Ferry, Florian Gallier, Simon Gonzalez, Nadège Lubin-Germain, Leandro Soter de Mariz E Miranda, et al.. Recent advances in the functionalization of unprotected carbohydrates. Amélia Pilar Rauter; Thisbe K Lindhorst; Yves Queneau. Carbohydrate Chemistry: Chemical and Biological Approaches, 45, Royal Society of Chemistry, pp.239-304, 2021, SPR - Carbohydrate Chemistry, 978-1-83916-390-6. ⟨10.1039/9781839164538-00239⟩. ⟨hal-03667486⟩
  • Benoit Crousse, Thierry Milcent. Synthesis of NCF3, NCF2H and NCH2CF3 motifs. merging Fluorinated Motifs. Properties, Synthesis and Applications, 2020. ⟨hal-03796648⟩
  • Danièle Bonnet-Delpon, Jean-Pierre Bégué, Benoit Crousse, Fabienne Grellepois, Constance Chollet, et al.. New 10-Trifluoromethyl Monomers, Dimers, and Chimeras of Artemisinin from a Key Allyl Bromide Precursor. Current fluoroorganic chemistry: new synthetic directions, technologies, materials and biological application, ACS Symposium Series, Vol 949, pp.337-351, 2007, ⟨10.1021/bk-2007-0949.ch020⟩. ⟨mnhn-02867458⟩
  • Jean-Hugues Renault, Jean-Marc Nuzillard, Olivier Intes, Alexandre Maciuk. Solvent systems. Alain Berthod. Comprehensive Analytical Chemistry Series, 38, Elsevier, pp.49-83, 2005, Countercurrent chromatography, the support-free liquid stationary phase, 978-0444507372. ⟨10.1016/S0166-526X(02)80006-X⟩. ⟨hal-01968195⟩

Brevets1 document

  • Maité Sylla-Iyarreta Veitía, Françoise Dumas, Georges Morgant. Synthesis Characterization and biological activities of metal-base complexes containing the leading drug valproic acid. France, Patent n° : PCT/FR2009/051077. 2009. ⟨hal-01487516⟩

Pré-publications, Documents de travail10 document

  • Yassine Mejri, Olivier Cailloux, Elvis Otogo N'Nang, Blandine Séon-Méniel, Jean-François Gallard, et al.. MS2DECIDE: Aggregating Multi-Annotated Tandem Mass Spectrometry Data with Decision Theory Enhances Natural Products Prioritization. 2025. ⟨hal-05058403⟩
  • Davide Di Lorenzo, Nicolo Bisi, Julia Kaffy, Lisa Marie Ramirez, Markus Zweckstetter, et al.. Synthetic chaperone based on Hsp90-Tau interaction inhibits pathological Tau aggregation and rescues physiological Tau-Microtubule interaction. 2025. ⟨hal-05047264⟩
  • Laurent Ferrié, Bruno Figadère, Nicolas Jamey, Bastien Champciaux. Peroxy-Carbenium Mediated Asymmetric Synthesis of 1,2-Dioxanes and 1,2-Dioxolanes. 2024. ⟨hal-04757792⟩
  • Florent Dumont, Emy Ponsardin, Guillaume Bernadat, Sylvia Cohen-Kaminsky. MOAL: Multi-Omic Analysis at Lab. A simplified methodology workflow to make reproducible omic bioanalysis. 2023. ⟨hal-04294241⟩
  • José Laxio Arenas, Jacopo Lesma, Tap Ha-Duong, Bikash Sahoo, Ayyalusamy Ramamoorthy, et al.. Relation between conformation and activity on islet amyloid polypeptide aggregation of fluorinated foldamers based on Ndifluoromethyl-1,4-triazole amino acids. 2023. ⟨hal-04273096⟩
  • Clémence Rose, Rodrigo Hernán Tomas-Grau, Brenda Zabala, Jean-Michel Brunel, Patrick Michel, et al.. Enhancing Inhibition of Both α-Synuclein Aggregation and Neuroinflammation: New Insights into the C-9 Modification of Doxycycline. 2023. ⟨hal-04250582⟩
  • Yazid Boutahri, Khoubaib Ben Haj Salah, Nicolas Tisserand, Nathalie Lensen, Benoit Crousse, et al.. Difluoroalanine: Synthesis, Incorporation in Peptides, and Hydrophobic Contribution Assessment. 2023. ⟨hal-04249424⟩
  • Mansour Dolé Kérim, Laurent Evanno, Laurent Ferrie. Stereodivergent Total Syntheses of (+)-Mycaperoxides C, D, G Methyl Ester and (-)-Mycaperoxide B. 2022. ⟨hal-03775643⟩
  • Marion Barthé, Flora Lefebvre, Emilie Langlois, Florence Lefebvre, Patrick Lechêne, et al.. PEGylated isoprenaline reveals distinct functions of cardiac β-adrenergic receptors located in the T-tubule vs . outer surface membrane. 2022. ⟨hal-03793970⟩
  • Damien Olivier-Jimenez, Zakaria Bouchouireb, Simon Ollivier, Julia Mocquard, Pierre-Marie Allard, et al.. From mass spectral features to molecules in molecular networks : a novel workflow for untargeted metabolomics. 2021. ⟨hal-05098952⟩

Thèses22 document

  • Sarah Szwarc. Développements méthodologiques en chimie analytique pour l'identification des enzymes catalysant des cyclisations C-N chez les alcaloïdes indolomonoterpéniques. Chimie analytique. Université Paris-Saclay, 2024. Français. ⟨NNT : 2024UPASQ074⟩. ⟨tel-05075853⟩
  • María Gutiérrez Sánchez. Macrophage Lysine Demethylase LSD1 : Implications for intracellular Leishmania survival and host-directed drug discovery.. Cell Behavior [q-bio.CB]. Université Paris-Saclay, 2023. English. ⟨NNT : 2023UPASQ042⟩. ⟨tel-04290331⟩
  • Kaliroi Peqini. Development of molecular probes acting on Tau/Tubulin and a-Synuclein/Tubulin interface. Medicinal Chemistry. Université Paris-Saclay; Università degli studi (Milan, Italie). Dipartimento di Scienze della Terra, 2023. English. ⟨NNT : 2023UPASQ036⟩. ⟨tel-04662379⟩
  • Mayssa Zayene. Conception, synthèse et valorisation biologique de nouveaux dérivés tropines et tropanes. Chimie organique. Université Paris-Saclay; Université de Monastir (Tunisie), 2023. Français. ⟨NNT : 2023UPASQ028⟩. ⟨tel-04639064⟩
  • Phuong Y Mai. Exploration ciblée de l'espace chimique des micro-organismes des « mares de kopara » polynésiennes. Chimie analytique. Université Paris-Saclay, 2023. Français. ⟨NNT : 2023UPASQ003⟩. ⟨tel-04536647⟩
  • Tingting Cao. Design and synthesis of new fluorinated hydrazines. Organic chemistry. Université Paris-Saclay, 2022. English. ⟨NNT : 2022UPASQ072⟩. ⟨tel-04058237⟩
  • Maxence Delaunay. Conception in silico d'inhibiteurs peptidiques d'interactions protéine-protéine. Bio-Informatique, Biologie Systémique [q-bio.QM]. Université Paris-Saclay, 2022. Français. ⟨NNT : 2022UPASQ069⟩. ⟨tel-04022527⟩
  • Zineb Fechtali Moute. Etude de la biodiversité et de la viabilité des amibes libres dans un réseau d'eau potable : approches environnementales et fondamentales. Parasitologie. Université Paris-Saclay, 2022. Français. ⟨NNT : 2022UPASQ062⟩. ⟨tel-04672721⟩
  • Chenghui Shi. Synthesis and conformational analysis of peptidomimetic foldamers containing diaza-peptide units : application in protein-protein interactions. Molecular biology. Université Paris-Saclay, 2022. English. ⟨NNT : 2022UPASQ055⟩. ⟨tel-04815486⟩
  • Ismaila Ciss. Synthèse totale des amphidinolides C et U. Chimie organique. Université Paris-Saclay; Université Cheikh Anta Diop (Dakar, Sénégal ; 1957-..), 2022. Français. ⟨NNT : 2022UPASQ039⟩. ⟨tel-04215937⟩
  • Mingxiang Zhu. New approaches to the synthesis of S/Se-glycosides and alkynyl C-nucleosides. Catalysis. Université Paris-Saclay, 2022. English. ⟨NNT : 2022UPASQ030⟩. ⟨tel-04153055⟩
  • Nedjwa Bennai. Étude de la réactivité des sucres dans les couplages organométalliques : application à la synthèse de glycosides biologiquement actifs. Chimie organique. Université Paris-Saclay; Université des Sciences et de la Technologie d'Oran Mohamed-Boudiaf (Algérie), 2022. Français. ⟨NNT : 2022UPASQ016⟩. ⟨tel-03681327⟩
  • Elodie Pradayrol. Vers la synthèse biomimétique de pigments fongiques : la sclérocitrine et la chalcitrine. Etude des métabolites de Scleroderma citrinum. Chimie organique. Université Paris-Saclay, 2022. Français. ⟨NNT : 2022UPASQ005⟩. ⟨tel-03662479⟩
  • José Laxio Arenas. Triazolamères fluorés : conception, synthèse, études conformationnelles et modulation de l'agrégation de peptides amyloïdes. Chimie thérapeutique. Université Paris-Saclay, 2022. Français. ⟨NNT : 2022UPASQ003⟩. ⟨tel-03962087⟩
  • Juba Ghouilem. Une nouvelle approche d'activation C(sp³) -H de sucres : vers de nouvelles classes de glycomimétiques C-hétérosides. Chimie organique. Université Paris-Saclay, 2021. Français. ⟨NNT : 2021UPASQ053⟩. ⟨tel-04334442⟩
  • Aminata Ouayogode. Etude ethnobotanique, chimique et activités pharmacologiques de plantes et recettes antimalariques de Côte d’Ivoire. Chimie thérapeutique. Université Paris-Saclay; Université Félix Houphouët-Boigny (Abidjan, Côte d'Ivoire), 2021. Français. ⟨NNT : 2021UPASQ034⟩. ⟨tel-03650772⟩
  • Sen Wang. Synthèse et fonctionnalisation d'azobenzènes : vers le développement de sondes photocommutables. Chimie organique. Université Paris-Saclay, 2021. Français. ⟨NNT : 2021UPASQ013⟩. ⟨tel-03341233⟩
  • Victor Turpin. Hypothèses de biosynthèse des alcaloïdes indolomonoterpéniques : résolution de mécanismes fondamentaux par la synthèse et par la modélisation. Chimie organique. Université Paris-Saclay, 2021. Français. ⟨NNT : 2021UPASQ009⟩. ⟨tel-03578052⟩
  • Jacopo Lesma. β-Hairpin peptidomimetics as inhibitors of hIAPP amyloid protein aggregation : design, synthesis and evaluation. Medicinal Chemistry. Université Paris-Saclay, 2020. English. ⟨NNT : 2020UPASQ018⟩. ⟨tel-03793799⟩
  • Siguara Bastos de Lemos E Silva. Chemistry and biosynthesis of highly complex marine alkaloids from Mediterranean biodiversity. Organic chemistry. Université Paris Saclay (COmUE), 2017. English. ⟨NNT : 2017SACLS214⟩. ⟨tel-02953258⟩
  • Elodie Jagu. Design, synthesis and biological evaluation of new polyamine derivatives as antikinetoplastid agents. Organic chemistry. Université Paris Saclay (COmUE), 2016. English. ⟨NNT : 2016SACLS589⟩. ⟨tel-01654426⟩
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