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Publications


735 documents

Journal articles629 document

  • Ping Gao, Xin Jiang, Jinyu Li, Julien Nicolas, Tâp Ha-Duong. Molecular Simulations of Polymer‐based Drug Nanocarriers: From Physical and Structural Properties to Controlled Release. Advanced Healthcare Materials, 2026, pp.e03503. ⟨10.1002/adhm.202503503⟩. ⟨hal-05459572⟩
  • Cảnh Hưng Nguyễn, Catherine Cailleau, Natalie Fournier, Luc Augis, Françoise Mercier-Nomé, et al.. Are hydrophilic deep eutectic solvents a potential vehicle for topical delivery of Amphotericin B against cutaneous leishmaniasis? An investigation of physicochemical properties, tolerability and antileishmanial efficacy. International Journal of Pharmaceutics, 2026, 689, pp.126439. ⟨10.1016/j.ijpharm.2025.126439⟩. ⟨hal-05397306⟩
  • Rany Mbeng Obame, Pierre Le Pogam, Karine Leblanc, Somia Rharrabti, Evodie Numbi Wa Ilunga, et al.. Targeted discovery of sesquiterpene indole alkaloids from Greenwayodendron suaveolens. Phytochemistry, 2026, 241, pp.114664. ⟨10.1016/j.phytochem.2025.114664⟩. ⟨hal-05327820⟩
  • Jonathan Sorres, Juliette Segret, Elsa Van-Elslande, David Touboul, Véronique Eparvier. Metabolomic analysis of macromycetes from French Guiana revueals chemodiversity in Xylariales order. Phytochemistry, 2026, 242, pp.114709. ⟨10.1016/j.phytochem.2025.114709⟩. ⟨hal-05333878⟩
  • Dario Cavaterra, Sara Giammaria, Irene Pandino, Gabriele Antonio Zingale, Valerio Delli Paoli, et al.. Citicoline Triggers Proteome Remodeling and Proteostatic Adaptation: Evidence from Shotgun Proteomics. Pharmaceutics, 2026, 18 (1), pp.61. ⟨10.3390/pharmaceutics18010061⟩. ⟨hal-05447472⟩
  • Flavio Alvarez, Florence Larrous, Ariel Mechaly, Benjamin Bardiaux, Quentin Goor, et al.. HTRF-based identification of small molecules targeting SARS-CoV-2 E protein interaction with ZO-1 PDZ2. Scientific Reports, In press, Online ahead of print. ⟨10.1038/s41598-025-31755-y⟩. ⟨hal-05449164⟩
  • Lucia Verrillo, Emiliano Manzo, Emma Cauzzi, Livia La Barbera, Giuseppina Sabatino, et al.. Microglial clearance, neuroprotection and cognitive recovery via a novel synthetic sulfolipid in Alzheimer’s disease. Journal of Neuroinflammation, 2025, ⟨10.1186/s12974-025-03634-w⟩. ⟨hal-05418674⟩
  • Grazia Raffaella Tundo, Gabriele Antonio Zingale, Irene Pandino, Elisa Peroni, Diego Sbardella, et al.. The Interplay Between the Ubiquitin–Proteasome System and Oxidative Stress: A Future Perspective in Eye Diseases. Antioxidants , 2025, 14 (12), pp.1475. ⟨10.3390/antiox14121475⟩. ⟨hal-05447475⟩
  • Khoubaib Ben Haj Salah, Elfried‐vannel Ngassam Ketchongue, Gabin Mwande-Maguene, Julien Pytkowicz. Fluorinated Bifunctional Iminophosphorane Organocatalysis (F‐BIMP): Application to Nitro‐Mannich Reaction. ChemistrySelect, 2025, 10 (45), pp.e06510. ⟨10.1002/slct.202506510⟩. ⟨hal-05398788⟩
  • Cagla Okyay, Jérôme Mathé, Nathalie Basdevant. Sequence and Force Effects on ssDNA Translocation through a Protein Nanopore: Coarse-Grained Steered Molecular Dynamics Simulations. Journal of Physical Chemistry B, 2025, ⟨10.26434/chemrxiv-2025-jz1v6⟩. ⟨hal-05396685⟩
  • George W P Madders, Marion Barthé, Flora Lefebvre, Emilie Langlois, Florence Lefebvre, et al.. Distinct functions of cardiac β-adrenergic receptors in the T-tubule vs. outer surface membrane. eLife, 2025, ⟨10.7554/eLife.84243⟩. ⟨hal-05273361⟩
  • Thais Santos, Eduardo Lages, Tiago Ricotta, Leandro de Oliveira, Guilherme Ramos, et al.. Long-Circulating Liposomes Codelivering Amphotericin B and Retinoic Acid for Cutaneous Leishmaniasis Treatment. ACS Omega, 2025, 10 (41), pp.48514-48530. ⟨10.1021/acsomega.5c06156⟩. ⟨hal-05302818⟩
  • Thierry Brigaud, Greta Varchi. Editorial: Recent advances in synthetic organic chemistry at the biomedical interface: honoring Professor Iwao Ojima on the occasion of his 80th birthday. Frontiers in Chemistry, 2025, 13, ⟨10.3389/fchem.2025.1721249⟩. ⟨hal-05325129⟩
  • Davide Di Lorenzo, Nicolo Bisi, Julia Kaffy, Lisa Marie Ramirez, Markus Zweckstetter, et al.. Synthetic chaperone based on Hsp90-Tau interaction inhibits Tau aggregation and rescues physiological Tau-Microtubule interaction. Nature Communications, 2025, 16 (1), pp.8756. ⟨10.1038/s41467-025-63824-1⟩. ⟨hal-05339048⟩
  • Soumaya Jemail, Emmanuel Magnier, Maxime Vitale, Guillaume Dagousset. Advances in Radical Remote γ-Functionalization of α,β-Unsaturated Carbonyl Compounds. Synthesis: Journal of Synthetic Organic Chemistry, 2025, ⟨10.1055/a-2705-6364⟩. ⟨hal-05364841⟩
  • George W. P. Madders, Marion Barthe, Flora Lefebvre, Emilie Langlois, Florence Lefebvre, et al.. Distinct functions of cardiac β-adrenergic receptors in the T-tubule vs. outer surface membrane. eLife, 2025, 14, pp.e84243. ⟨hal-05271952⟩
  • Dimitra Kyrko, Tingting Cao, Pascal Retailleau, Julia Kaffy, Benoît Crousse. Access to N -Fluorinated Azapeptides and Azapeptoids as Peptidomimetic Scaffolds. ACS Organic & Inorganic Au, 2025, ⟨10.1021/acsorginorgau.5c00073⟩. ⟨hal-05248269⟩
  • Alice Vetrano, Nico Di Fonte, Olivier Monasson, Federico Perrella, Martina Porco, et al.. Enantiopurity-Dependent Peptide Coacervates and Asymmetric Organocatalysis. BioRxiv, 2025, ⟨10.1101/2025.08.13.670095⟩. ⟨hal-05345892⟩
  • Nalia Mekarnia, Sandrine Cojean, Philippe Loiseau. Resistance to Antileishmanial Drug Candidates: A Flowchart for an Early Phenotypic Evaluation of Risk. Drugs and Drug Candidates, 2025, 4 (3), pp.38. ⟨10.3390/ddc4030038⟩. ⟨hal-05235475⟩
  • Farzin Arjmand, Elisa Peroni, Michel Boissiere, Adrien Mourgout, Aazedine Lamouri, et al.. Corrosion inhibition by grafted nitrophenyl and BMP-2 peptide derivatives on a Ti 35 Zr 25 Nb 25 (MoTa) 15 high-entropy alloy. Corrosion Engineering, Science and Technology, 2025, ⟨10.1177/1478422X251358647⟩. ⟨hal-05345865⟩
  • Quentin Joachim, Delphine Carry, Mattéo Di Pasquale, Jérôme Marrot, Suzuka Yamamoto, et al.. Introduction of Structural Diversity at the C2 Position of Unsaturated Iminosugars through Palladium‐Catalyzed Cross‐Coupling Reactions. European Journal of Organic Chemistry, 2025, 28 (32), ⟨10.1002/ejoc.202500502⟩. ⟨hal-05326462⟩
  • Alessia Distefano, Paolo Corsaro, Nunzio Tuccitto, Francesca Laneri, Olivier Monasson, et al.. Intrinsically photoluminescent hydrogels to measure peptides‑copper binding affinities. Journal of Inorganic Biochemistry, 2025, 268, pp.112914. ⟨10.1016/j.jinorgbio.2025.112914⟩. ⟨hal-05052019⟩
  • Mayssa Zayene, Franck Le Bideau, Pascal Retailleau, Hichem Ben Jannet, Vincent Gandon, et al.. Dual Photoredox/Cu‐Catalysis Enables Diastereoselective Synthesis of 3‐ β ‐Ethynyltropanes via Decarboxylative Alkynylation. Advanced Synthesis and Catalysis, 2025, ⟨10.1002/adsc.202500241⟩. ⟨hal-05114385⟩
  • Zina Benissa, Fatma Chtourou, Françoise Dumas, Sylvie Bouttier, Mohamed Bouaziz, et al.. Chemometric study of the effects of the geographical origin and the collection period on the chemical compositions and the antimicrobial activities of Pituranthos tortuosus essential oils. Zeitschrift fur Naturforschung C, 2025, ⟨10.1515/znc-2024-0302⟩. ⟨hal-05192588⟩
  • Lhana Tisseur, Cédric Logé, Sandrine Cojean, Khadidiatou Gassama, Lilian Karcher, et al.. Pharmacophore-guided optimization of the hit compound CTN1122 in the design of promising imidazo[1,2- a ]pyrazine derivatives targeting the casein kinase 1 for antileishmanial therapy. RSC Medicinal Chemistry, In press, ⟨10.1039/d5md00257e⟩. ⟨hal-05173262⟩
  • Ömer Taspinar, Daniel J Leonard, Nathan Picois, Cornelia Göcke, Matej Žabka, et al.. Asymmetric Intramolecular α‐Arylation of Polar Amino Acids Bearing β‐Leaving Groups. Angewandte Chemie International Edition, 2025, ⟨10.1002/anie.202507713⟩. ⟨hal-05110334⟩
  • Sarah Szwarc, Adriano Rutz, Kyungha Lee, Yassine Mejri, Olivier Bonnet, et al.. Translating community-wide spectral library into actionable chemical knowledge: a proof of concept with monoterpene indole alkaloids. Journal of Cheminformatics, 2025, 17, pp.62. ⟨10.1186/s13321-025-01009-0⟩. ⟨hal-05058394⟩
  • Xinya Liu, Valentin Dorokhov, Olivier Provot, Christine Tran, Pascal Retailleau, et al.. Mechanochemical Approach for Metal‐Free Regioselective C5‐Sulfenylation of Imidazo[2,1‐b]thiazoles. ChemSusChem, 2025, ⟨10.1002/cssc.202500320⟩. ⟨hal-05053681⟩
  • Ellen Gonçalves De Oliveira, Juliane Sousa Lanza, Sandrine Cojean, Paulo Otávio L. Moreira, Luiza Guimarães Tunes, et al.. Re-sensitization of antimony-resistant Leishmania by highly potent SbV-porphyrin through the involvement of ERG6-coding gene. Biomedicine and Pharmacotherapy, 2025, 187, pp.118059. ⟨10.1016/j.biopha.2025.118059⟩. ⟨hal-05445980⟩
  • Jun Yan, Pascal Retailleau, Abdallah Hamze, Christine Tran. Copper‐Catalyzed Domino Synthesis of Spiropyrazoline Oxindoles via Condensation of Indolin‐2‐One and Phenylhydrazine Derivatives. Advanced Synthesis and Catalysis, 2025, 367 (10), ⟨10.1002/adsc.202500223⟩. ⟨hal-05127035⟩
  • Moussa Touré, Abdoulaye Gassama, Oumar Sambou, Christian Cavé, Sandrine Cojean. Synthesis and in vitro/in silico evaluation of the antimalarial activity of potential amino-quinoline derivatives. European Journal of Medicinal Chemistry Reports, 2025, 13, pp.100241. ⟨10.1016/j.ejmcr.2024.100241⟩. ⟨hal-05445961⟩
  • Davide Di Lorenzo, Nicolo Bisi, Raffaella Bucci, Inga Ennen, Leonardo Lo Presti, et al.. Application of modular isoxazoline-β$^{2,2-}$amino acid-based peptidomimetics as chemical model systems for studying the tau misfolding. iScience, 2025, 28 (4), pp.112272. ⟨10.1016/j.isci.2025.112272⟩. ⟨hal-05056022⟩
  • Florent Edde, Emmanuelle Drège, Laurent Evanno. User‐friendly and Green Procedure for a Photoinduced Wohl‐Ziegler Reaction. European Journal of Organic Chemistry, 2025, 28 (18), ⟨10.1002/ejoc.202500183⟩. ⟨hal-05114321⟩
  • Mathew Choaji, Ascel Samba-Louaka, Zineb Fechtali-Moute, Willy Aucher, Sébastien Pomel. Encystment and Excystment Processes in Acanthamoeba castellanii: An Emphasis on Cellulose Involvement. Pathogens, 2025, 14, ⟨10.3390/pathogens14030268⟩. ⟨hal-04988818⟩
  • Mohamed Belemlilga, Hazrina Hazni, Aristide Traore, Indira Dennemont, Sébastien Pomel, et al.. Chemical analysis by molecular networking methods on extracts of Saba senegalensis (A.DC.) Pichon (Apocynaceae) and its anthelmintic activity on Caenorhabditis elegans. Clinical Traditional Medicine and Pharmacology, 2025, 6 (1), pp.200195. ⟨10.1016/j.ctmp.2025.200195⟩. ⟨hal-05149228⟩
  • Angélique Ferry. Diversity in glycochemistry through metal-catalyzed reactions. Comptes Rendus. Chimie, 2025, 28 (G1), pp.199-213. ⟨10.5802/crchim.373⟩. ⟨hal-05349682⟩
  • Shashank Pandey, Elisa Peroni, Dagmar Jarkovska, Magdalena Chottova Dvorakova, Olivier Monasson, et al.. Role of Neuropeptide B/W Signaling in Modulating Intracellular Calcium in Human Skin Fibroblasts. Frontiers in Bioscience-Landmark, 2025, 30 (2), ⟨10.31083/FBL26760⟩. ⟨hal-04971764⟩
  • Alicia Maroto, Olivier Briand, Alessia Distefano, Filiz Arioz, Olivier Monasson, et al.. Differentiation of Isomeric TAT1-CARNOSINE Peptides by Energy-Resolved Mass Spectrometry and Principal Component Analysis. Molecules, 2025, Special Issue Design, Synthesis, and Analysis of Potential Drugs, 3rd Edition, 30 (4), pp.853. ⟨10.3390/molecules30040853⟩. ⟨hal-04943837⟩
  • Marion Alter, Margherita Donnici, Solenn Reguer, Mathieu Thoury, Matthieu Réfrégiers, et al.. Alteration markers of green copper bimetallic pigments in easel paintings by an inter-comparison of analogues and historical samples. Microchemical Journal, 2025, 209, pp.112541. ⟨10.1016/j.microc.2024.112541⟩. ⟨hal-04942544⟩
  • Alexandra Bordes, Isabelle Opalinski, Fabien Thoreau, Olivier Provot, Abdallah Hamze, et al.. β-Glucuronidase-Responsive Albumin-Binding Prodrug of Colchicine-Site Binders for Selective cancer Therapy. ChemMedChem, 2025, 20 (9), pp.e202400969. ⟨10.1002/cmdc.202400969⟩. ⟨hal-04918349⟩
  • Monika Skibinska, Alicja Warowicka, Benoît Crousse, Tomasz Cytlak. Synthesis and Antibacterial Activity of Novel Phosphonated CF3-β-lactams. ACS Omega, 2025, 10 (17), pp.18062-18072. ⟨10.1021/acsomega.5c01562⟩. ⟨hal-05105385⟩
  • Lorenzo Meneghelli, Stephanie Davidson, Anthony Gineste, Lamia El Guermah, Sabrina Kellouche-Gaillard, et al.. Design and synthesis of a clickable cell-permeable pseudopeptide Pin1 inhibitor with antiproliferative effects on human multiple myeloma cell line. Chemical Communications, 2025, ⟨10.1039/D4CC05968A⟩. ⟨hal-05003977⟩
  • Thaís Antonia Alves Fernandes, Aurore Tourville, Ismaila Ciss, Rafaela Ribeiro Silva, Bianca Andretto de Mattos, et al.. Oxytetracycline and its Non-Antibiotic Derivative DOT Protect Midbrain Dopamine Neurons from Iron-Driven Oxidative Damage. Neurotoxicity Research, 2025, 43 (2), pp.16. ⟨10.1007/s12640-025-00742-6⟩. ⟨hal-05190872⟩
  • Yingmin Jiang, Tâp Ha-Duong. Temperature-Dependent Coarse-Grained Model for Simulations of Intrinsically Disordered Protein LCST and UCST Liquid–Liquid Phase Separations. Journal of Chemical Theory and Computation, 2025, 21 (9), pp.4939-4952. ⟨10.1021/acs.jctc.5c00212⟩. ⟨hal-05373622⟩
  • Louis-Valentin Méteignier, Sarah Szwarc, Patra Barunava, Mickael Durand, Duchesse-Lacours Zamar, et al.. Harnessing the spatial and transcriptional regulation of monoterpenoid indole alkaloid metabolism in Alstonia scholaris leads to the identification of broad geissoschizine cyclase activities. Plant Physiology and Biochemistry, 2025, 219, pp.109363. ⟨10.1016/j.plaphy.2024.109363⟩. ⟨hal-04810555⟩
  • Ahmed El Rhaz, Lisa Bonin, Ameni Hadj Mohamed, Samir Messaoudi. Advances in metal-catalyzed strategies for carbohydrate functionalization. Chemical Communications, 2025, 61 (84), pp.16331-16353. ⟨10.1039/D5CC04316F⟩. ⟨hal-05443477⟩
  • Rany B. Mbeng Obame, Sidney Gallard, Sacha Gibert, Jean-François Gallard, Solenn Ferron, et al.. Unifying the Absolute Configuration of Dibenzopyrrocoline Alkaloids with Relative Configuration Revision of Cryptowolinol and Description of Isocryptaustoline from Cryptocarya oubatchensis. Journal of Natural Products, 2025, ⟨10.1021/acs.jnatprod.4c01315⟩. ⟨hal-05024657⟩
  • Bastien Champciaux, Nicolas Jamey, Bruno Figadère, Laurent Ferrié. Peroxycarbenium-Mediated Asymmetric Synthesis of 1,2-Dioxanes and 1,2-Dioxolanes. Journal of the American Chemical Society, 2025, 147 (4), pp.3353-3359. ⟨10.1021/jacs.4c13899⟩. ⟨hal-04918894⟩
  • Yassine Mejri, Olivier Cailloux, Elvis Otogo N’nang, Blandine Séon-Méniel, Jean‐françois Gallard, et al.. MS2DECIDE: Aggregating Multiannotated Tandem Mass Spectrometry Data with Decision Theory Enhances Natural Products Prioritization. Chemistry–Methods, In press, ⟨10.1002/cmtd.202400088⟩. ⟨hal-05286889⟩
  • Laurent Ferrié. Les endoperoxydes, des hétérocycles singuliers. L'Actualité Chimique, 2025, 505, pp.21-27. ⟨hal-05346766⟩
  • Yuqing Zhang, Myriam Eveno, Nadège Lubin-Germain, Agnès Lattuati-Derieux, Nadège Lubin-Germain, et al.. Partially fluorinated derivatives as a powerful tool for the restoration of blanched easel paintings. Progress in Organic Coatings, 2025, 207, pp.109375. ⟨10.1016/j.porgcoat.2025.109375⟩. ⟨hal-05104320⟩
  • Makiath Adebo, Mathilda Bonnet, Ons Laouej, Celine Defaix, Josephine C. Mcgowan, et al.. Psilocybin as Transformative Fast‐Acting Antidepressant : Pharmacological Properties and Molecular Mechanisms. Fundamental & Clinical Pharmacology, 2025, 39 (4), pp.e70038. ⟨10.1111/fcp.70038⟩. ⟨hal-05237520⟩
  • Marceau Levasseur, Alice Trac, Isabelle Clavereau, Flavien Zannini, Yannick Estevez, et al.. Reverse chemical ecology to study the defense of the plant host Sextonia rubra and the chemical mediators of its endophyte Fusarium falciforme against phytopathogen Trametes versicolor. Phytochemistry, 2025, 238, pp.114577. ⟨10.1016/j.phytochem.2025.114577⟩. ⟨hal-05128635⟩
  • Ahmed El Rhaz, Estelle Messé, Pascal Retailleau, William Erb, Samir Messaoudi, et al.. Access to Thioglycoconjugate Bioorganometallic Ferrocenes via a Copper-Catalyzed Coupling. Organic Letters, 2025, 27 (29), pp.7979-7985. ⟨10.1021/acs.orglett.5c02292⟩. ⟨hal-05222831⟩
  • Bartosz Godlewski, Nina Bozinovic, Quentin Joachim, Olivier Monasson, Nadège Lubin-Germain, et al.. Direct palladium-catalyzed C–H arylation of bioactive triazolyl- C -nucleosides on a key position of the heterocyclic base. Chemical Communications, 2025, 61 (85), pp.16584-16587. ⟨10.1039/D5CC04215A⟩. ⟨hal-05349690⟩
  • Bianca Andretto de Mattos, Rodrigo Hernán Tomas-Grau, Thaís Antonia Alves Fernandes, Florencia González-Lizárraga, Aurore Tourville, et al.. Uric Acid, the End-Product of Purine Metabolism, Mitigates Tau-Related Abnormalities: Comparison with DOT, a Non-Antibiotic Oxytetracycline Derivative. Biomolecules, 2025, 15 (7), pp.941. ⟨10.3390/biom15070941⟩. ⟨hal-05346486⟩
  • Farzin Arjmand, Alima Chali, Youssef Snoussi, David Troadec, Gilles Patriarche, et al.. In-situ chemical grafting of aminophenyl and RGD peptide on an equimolar high-entropy HfNbTaTiZr alloy: electrochemical behavior and surface characterization. Emergent Materials, 2024, ⟨10.1007/s42247-024-00963-z⟩. ⟨hal-04854358⟩
  • Norbert Hoffmann, Mario Andrés Gomez Fernandez, Arthur Desvals, Corentin Lefebvre, Clément Michelin, et al.. Photochemical reactions of biomass derived platform chemicals. Frontiers in Chemistry, 2024, 12, ⟨10.3389/fchem.2024.1485354⟩. ⟨hal-04831095⟩
  • Carlos dos Santos, Daniel Silva, Julie Le Bescont, Chloé Breton-Patient, Sandrine Piguel, et al.. Studying the influence of electron donor-withdraw groups on the photophysical properties of 3-arylthioimidazo[1,2- a ]pyridines: experimental and theoretical study. Molecular Physics, 2024, 123 (14), e2436625 (13 p.). ⟨10.1080/00268976.2024.2436625⟩. ⟨hal-05261891⟩
  • Thierry Milcent, Pascal Retailleau, Benoit Crousse, Sandrine Ongeri. Synthesis of extended fluorinated tripeptides based on the tetrahydropyridazine scaffold. Beilstein Journal of Organic Chemistry, 2024, 20, pp.3174-3181. ⟨10.3762/bjoc.20.262⟩. ⟨hal-05142142⟩
  • Julien Pytkowicz, Grégory Chaume, Nathalie Lensen, Evelyne Chelain, Thierry Brigaud. Two decades of fluorine chemistry in Cergy. Comptes Rendus. Chimie, 2024, 27 (G1), pp.353-383. ⟨10.5802/crchim.360⟩. ⟨hal-04823676⟩
  • Sarah Szwarc, Pierre Le Pogam, Mehdi Beniddir. Emerging trends in plant natural products biosynthesis: a chemical perspective. Current Opinion in Plant Biology, 2024, 82, pp.102649. ⟨10.1016/j.pbi.2024.102649⟩. ⟨hal-05058399⟩
  • Abda Ba, Vincent Roumy, Malak Al Ibrahim, Kristelle Hughes, Thierry Hennebelle, et al.. Antileishmanial, antitrypanosomal and anti-coronavirus activities of benzophenanthridine alkaloids and other specialized metabolites isolated from the root bark of Zanthoxylum zanthoxyloides (Lam.) B.Zepernick & Timler. Fitoterapia, 2024, 179, pp.106232. ⟨10.1016/j.fitote.2024.106232⟩. ⟨hal-05349457⟩
  • Sakna Bazzi, Ameni Hadj Mohamed, Dmytro Ryzhakov, Juba Ghouilem, Mehdi Beniddir, et al.. Diastereoselective Anomeric C(sp 3 )−H Cyclization Towards the Design of New Cyclophane‐Braced Glycopeptides. Angewandte Chemie International Edition, 2024, 64 (6), ⟨10.1002/anie.202418057⟩. ⟨hal-05418610⟩
  • Enzo Lezin, Mickael Durand, Caroline Birer Williams, Ana Luisa Lopez Vazquez, Thomas Perrot, et al.. Genome‐based discovery of pachysiphine synthases in Tabernaemontana elegans. The Plant Journal, 2024, 120 (5), pp.1880-1900. ⟨10.1111/tpj.17085⟩. ⟨hal-05036872⟩
  • Gulsah Bayraktar, Pascal Marchand, Euzébio Guimarães Barbosa, Marilia Cecilia da Silva, Karen Cacilda Weber, et al.. Biological properties and in silico studies of thiazolopyrimidine derivatives active against visceral and cutaneous Leishmania spp. amastigote forms. European Journal of Medicinal Chemistry Reports, 2024, 12, pp.100228. ⟨10.1016/j.ejmcr.2024.100228⟩. ⟨hal-05088062⟩
  • Linlin Li, Emma Lemouton, Yahya Al Ayi, Dmytro Ryzhakov, Pascal Retailleau, et al.. Expanding 1‐Aminosugar Synthesis through Activated Glycals’ Reactivity. European Journal of Organic Chemistry, 2024, 27 (41), ⟨10.1002/ejoc.202400728⟩. ⟨hal-05349640⟩
  • Aurélie Honfroy, Jolien Bertouille, Ana-Maria Turea, Thibault Cauwenbergh, Jessica Bridoux, et al.. Fluorinated Peptide Hydrogels Result in Longer In Vivo Residence Time after Subcutaneous Administration. Biomacromolecules, 2024, 25 (10), pp.6666-6680. ⟨10.1021/acs.biomac.4c00872⟩. ⟨hal-04782661⟩
  • Nalia Mekarnia, Kamal-Eddine Benallal, Jovana Sádlová, Barbora Vojtková, Aurélie Mauras, et al.. Effect of Phlebotomus papatasi on the fitness, infectivity and antimony-resistance phenotype of antimony-resistant Leishmania major Mon-25. International journal for parasitology. Drugs and drug resistance, 2024, 25, pp.100554. ⟨10.1016/j.ijpddr.2024.100554⟩. ⟨hal-04632483⟩
  • Pieter Langerhorst, Melissa Baerenfaenger, Purva Kulkarni, Simon Nadal, Charissa Wijnands, et al.. N-linked glycosylation of the M-protein variable region: glycoproteogenomics reveals a new layer of personalized complexity in multiple myeloma. Clinical Chemistry and Laboratory Medicine, 2024, 62 (8), pp.1626-1635. ⟨10.1515/cclm-2023-1189⟩. ⟨hal-05085563⟩
  • Dimitra Kyrko, Murat Saraç, Jing Hao, Pascal Retailleau, Sandrine Ongeri, et al.. Functionalized α‐Fluorinated Amines from Imines and Enol Ethers. Advanced Synthesis and Catalysis, 2024, 366 (16), pp.3460-3465. ⟨10.1002/adsc.202400517⟩. ⟨hal-04756974⟩
  • Farzin Arjmand, Adrien Mourgout, Alima Chali, Madjid Djemai, Credson-Yannick Langueh, et al.. L-PBF processing and characterization of a Ti 35 Nb 30 Zr 29 Mo 3 Ta 3 multiprincipal element alloy for medical implants. Applied Physics Letters, 2024, 125 (4), pp.041904. ⟨10.1063/5.0208341⟩. ⟨hal-04739764⟩
  • Milene Hornink, Monica Toledo, Daniel Pimenta, Caio Paschoalin, Pamela Silva, et al.. 1-Iodoglycal: A Versatile Intermediate for the Synthesis of d -Glyco Amides and Esters Employing Carbonylative Cross-Coupling Reaction. ACS Omega, 2024, 9 (29), pp.31732-31744. ⟨10.1021/acsomega.4c02645⟩. ⟨hal-05349644⟩
  • Yu Fan, Ahmed El Rhaz, Stéphane Maisonneuve, Emilie Gillon, Maha Fatthalla, et al.. Photoswitchable glycoligands targeting Pseudomonas aeruginosa LecA. Beilstein Journal of Organic Chemistry, 2024, 20, pp.1486-1496. ⟨10.3762/bjoc.20.132⟩. ⟨hal-04637573⟩
  • Nicolas Jamey, Laurent Ferrié. Stereodivergent Total Synthesis of Ethyl Plakortide Z. Organic Letters, 2024, 26 (27), pp.5741-5745. ⟨10.1021/acs.orglett.4c01893⟩. ⟨hal-04738657⟩
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  • Maité Iyarreta Veitia Sylla-Iyarreta Veitía, Françoise Dumas, Georges Morgant, Yves Frapart, Alain Tomas, et al.. Synthesis, structural analysis and anticonvulsant activity of a ternary Cu (II) mononuclear complex containing 1, 10-phenanthroline and the leading antiepileptic drug valproic acid. Biochimie, 2009, 91 (10), pp.1286-1293. ⟨10.1016/j.biochi.2009.06.015⟩. ⟨hal-01487475⟩
  • Daniela Vuluga, Julien Legros, Benoit Crousse, Danièle Bonnet-Delpon. Synthesis of pyrazoles through catalyst-free cycloaddition of diazo compounds to alkynes. Green Chemistry, 2009, 11 (2), pp.156-159. ⟨10.1039/B812242C⟩. ⟨hal-02326141⟩
  • Abdallah Hamze, Anne Giraud, Samir Messaoudi, Olivier Provot, Jean-François Peyrat, et al.. Synthesis, Biological Evaluation of 1,1-Diarylethylenes as a Novel Class of Antimitotic Agents. ChemMedChem, 2009, 4 (11), pp.1912-1924. ⟨10.1002/cmdc.200900290⟩. ⟨hal-02394586⟩
  • Jean-Daniel Brion, Mouad Alami, Bret Tréguier, Abdallah Hamze, Olivier Provot. Expeditious synthesis of 1,1-diarylethylenes related to isocombretastatin A-4 (isoCA-4) via palladium-catalyzed arylation of N-tosylhydrazones with aryl triflates. Tetrahedron Letters, 2009, 50 (47), pp.6549-6552. ⟨10.1016/j.tetlet.2009.09.046⟩. ⟨hal-02394584⟩
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  • Céline Mousset, Olivier Provot, Abdallah Hamze, Jérôme Bignon, Jean-Daniel Brion, et al.. DMSO–PdI2 as a powerful oxidizing couple of alkynes into benzils: one-pot synthesis of nitrogen-containing five- or six-membered heterocycles. Tetrahedron, 2008, 64 (19), pp.4287-4294. ⟨10.1016/j.tet.2008.02.081⟩. ⟨hal-02394600⟩
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  • Anne Giraud, Olivier Provot, Abdallah Hamze, Jean-Daniel Brion, Mouad Alami. One-pot hydrosilylation–protodesilylation of functionalized diarylalkynes: a highly selective access to Z-stilbenes. Application to the synthesis of combretastatin A-4. Tetrahedron Letters, 2008, 49 (7), pp.1107-1110. ⟨10.1016/j.tetlet.2007.12.057⟩. ⟨hal-02394604⟩
  • Céline Mousset, Anne Giraud, Olivier Provot, Abdallah Hamze, Jérôme Bignon, et al.. Synthesis and antitumor activity of benzils related to combretastatin A-4. Bioorganic and Medicinal Chemistry Letters, 2008, 18 (11), pp.3266-3271. ⟨10.1016/j.bmcl.2008.04.053⟩. ⟨hal-02394592⟩
  • Daniela Vuluga, Julien Legros, Benoit Crousse, Danièle Bonnet-Delpon. Solubility switch of gold nanoparticles through hydrogen bond association. Chemical Communications, 2008, 40, pp.4954. ⟨10.1039/b810932j⟩. ⟨hal-02326146⟩
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  • J. d'Angelo, G. Morgant, N.E. Ghermani, D. Desmaele, B. Fraisse, et al.. Crystal structures and physico-chemical properties of Zn(II) and Co(II) tetraaqua(3-nitro-4-hydroxybenzoato) complexes: their anticonvulsant activities as well as related (5-nitrosalicylato)-metal complexe. Polyhedron, 2008, 27 (2), pp.537-546. ⟨10.1016/j.poly.2007.10.006⟩. ⟨hal-00382739⟩
  • Gaëlle Le Bras, Abdallah Hamze, Samir Messaoudi, Olivier Provot, Pierre-Benoît Le Calvez, et al.. Synthesis of Isocoumarin via PTSA-Catalyzed Annulation of Diarylalkynes. Synthesis: Journal of Synthetic Organic Chemistry, 2008, 2008 (10), pp.1607-1611. ⟨10.1055/s-2008-1072575⟩. ⟨hal-02394596⟩
  • N.E. Ghermani, G. Morgant, J. d'Angelo, D. Desmaele, B. Fraisse, et al.. Covalently bonded infinite zigzag chain structure in a novel Zn(II) complex of 2.5-dihydroxy-1.6-benzenedicarboxylic acid. Polyhedron, 2007, 26 (12), pp.2880-2884. ⟨10.1016/j.poly.2007.01.025⟩. ⟨hal-00382749⟩
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  • Gaëlle Le Bras, Olivier Provot, Jean-François Peyrat, Mouad Alami, Jean-Daniel Brion. Rapid microwave assisted hydration of internal arylalkynes in the presence of PTSA: an efficient regioselective access to carbonyl compounds. Tetrahedron Letters, 2006, 47 (31), pp.5497-5501. ⟨10.1016/j.tetlet.2006.05.155⟩. ⟨hal-02394618⟩
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  • Anne Giraud, Olivier Provot, Jean-François Peyrat, Mouad Alami, Jean-Daniel Brion. Microwave-assisted efficient synthesis of 1,2-diaryldiketones: a novel oxidation reaction of diarylalkynes with DMSO promoted by FeBr3. Tetrahedron, 2006, 62 (33), pp.7667-7673. ⟨10.1016/j.tet.2006.05.072⟩. ⟨hal-02394615⟩
  • A. Fourneret-Vivier, B. Lebeau, M. R. Mallaret, M. P. Brenier-Pinchart, J. P. Brion, et al.. Hospital-wide prospective mandatory surveillance of invasive aspergillosis in a French teaching hospital (2000-2002).. Journal of Hospital Infection, 2006, 62 (1), pp.22-8. ⟨10.1016/j.jhin.2005.06.013⟩. ⟨hal-00171251⟩
  • Nathalie L'Hermite, Anne Giraud, Olivier Provot, Jean-François Peyrat, Mouad Alami, et al.. Disproportionation reaction of diarylcarbinols: a versatile access to diarylmethanes speeded up using microwave irradiation. Tetrahedron, 2006, 62 (51), pp.11994-12002. ⟨10.1016/j.tet.2006.09.083⟩. ⟨hal-02394612⟩
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  • Alexandre Maciuk, Jean-Hugues Renault, Rodolphe Margraff, Philippe Trébuchet, Monique Zeches-Hanrot, et al.. Anion-Exchange Displacement Centrifugal Partition Chromatography. Analytical Chemistry, 2004, 76 (21), pp.6179-6186. ⟨10.1021/ac049499w⟩. ⟨hal-01968198⟩
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  • Abdelkhaleq Legssyer, Hassane Mekhfi, Mohamed Bnouham, Vincent Roumy, Christine Herrenknecht, et al.. Tannins and catechin gallate mediate the vasorelaxant effect of Arbutus unedo on the rat isolated aorta. Phytotherapy Research, 2004, 18 (11), pp.889-894. ⟨10.1002/ptr.1513⟩. ⟨hal-03161416⟩
  • M. Pizzonero, L. Keller, F. Dumas, M. Ourevitch, G. Morgant, et al.. Crystallographic/experimental electron density characterizations and reactions with nucleophiles of β-enaminonitriles possessing a pyrrolobenzazepine core. Journal of Organic Chemistry, 2004, 69 (13), pp.4336-4350. ⟨10.1021/jo049681x⟩. ⟨hal-02296123⟩
  • Jean-François Berrien, Olivier Provot, Joëlle Mayrargue, Michel Coquillay, Liliane Cicéron, et al.. Alkylation of manganese(ii) tetraphenylporphyrin by a synthetic antimalarial trioxane. Organic & Biomolecular Chemistry, 2003, 1 (16), pp.2859. ⟨10.1039/b302835f⟩. ⟨hal-02394634⟩
  • Laure Cointeaux, Jean-François Berrien, Viviane Peyrou, Olivier Provot, Liliane Cicéron, et al.. Synthesis and antimalarial activity of 2-methoxyprop-2-yl peroxides derivatives. Bioorganic and Medicinal Chemistry Letters, 2003, 13 (1), pp.75-77. ⟨10.1016/S0960-894X(02)00837-5⟩. ⟨hal-02394637⟩
  • Cécile Pégurier, Laurence Morellato, Eminn Chahed, Jean Andrieux, Jean Paul Nicolas, et al.. Synthesis of new arylalkoxy amido derivatives as melatoninergic ligands.. Bioorganic and Medicinal Chemistry, 2003, 11-5 (5), pp.789-800. ⟨10.1016/s0968-0896(02)00328-0⟩. ⟨hal-00080328⟩
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  • Florian Malard, Eric Jacquet, Naima Nhiri, Christina Sizun, Amélie Chabrier, et al.. Atomic level description of the Binding of the Cancer-Related TCTP Protein to the sertraline drug and to the anti-apoptotic Mcl-1 protein. Biotechnocentre, Biotechnocentre, Oct 2021, Chaumont sur Tharonne, France. ⟨hal-04396389⟩
  • David Montoir, Mehdi Amoura, Zine El Abidine Ababsa, T.M. Vishwanatha, Expédite Yen-Pon, et al.. Synthesis of aryl-thioglycopeptides through chemoselective Pd-mediated conjugation. 4. GFPP Chemical Ligation Meeting (Ligation2020), Jan 2020, Orléans, France. ⟨hal-02892772⟩
  • Lucile Brunel-Duverger, Caroline Thomas, Noelle Timbart. « Ateliers, groupes techniques et mains d'artistes : les cercueils à fond jaune de la Troisième Période intermédiaire ». Le Centre de Recherche et de Restauration des Musées de France : 20 ans déjà !, actes du colloque à la Cité de l’Architecture et du Patrimoine, Paris, 20 novembre 2019, L. Mailho, M. Menu, Nov 2019, Paris, France. publication en ligne du C2RMF, 2021 : https://c2rmf.fr/journees-detudes-du-c2rmf, p. 107-117. ⟨hal-03745088⟩
  • Oumayma Hamzaoui, Alexandre Maciuk, Sabine Delgrange, Katia Kerdja, Claire Thouminot, et al.. Cannalactone: a new non-canonical strigolactone exudated by Cannabis sativa roots with a pivotal role in host specialization within French broomrape (Phelipanche ramosa) populations. 15th World Congress on Parasitic Plants, Jun 2019, Amsterdam, Netherlands. ⟨hal-02326484⟩
  • D. Touboul, L. Laboureur, H. Thi Phuong Thuy, P. Champy, V. Eparvier. Supercritical fluid chromatography coupled to high resolution mass spectrometry for dereplication and quantification of natural products. RFMF, May 2019, Clermond - Ferrand, France. ⟨hal-04410154⟩
  • Bastien Nay, Erwan Poupon. La recherche en synthèse biomimétique. Journées Convergence CNRS en Synthèse Totale de Molécules Complexes, Jan 2019, Nantes, France. ⟨hal-04303748⟩
  • Emeric Miclet, Anas Terrien, Claire Loison, Luminita Duma, Thierry Brigaud, et al.. New insights into the structural and dynamics properties of collagen model peptides using CD spectroscopy, MD simulations and innovative NMR approaches. 35th European Peptide Symposium, Aug 2018, Dublin, Ireland. pp.192-194, ⟨10.17952/35EPS.2018.192⟩. ⟨hal-02057961⟩
  • Sandrine Pagès-Camagna, Lucile Brunel-Duverger, Christel Doublet, Eric Laval, Nancy Brodie-Linder, et al.. Contribution from SEM Studies in the Understanding of Degradation Mechanisms of Copper Green Pigments from the Louvre Museum’s 21st Dynasty Egyptian Coffins. Microscopy & Microanalysis 2018 Meeting, Aug 2018, Baltimore, MD, United States. pp.2126-2127, ⟨10.1017/S143192761801111X⟩. ⟨hal-01867962⟩
  • Marion Alter, Anne-Solenn Le Hô, Ludovic Bellot-Gurlet, Céline Paris, Margherita Donnici, et al.. Alteration of green copper-based organometallic pigments: influence of the organic matrix on the chromatic modification. E-MRS Spring Meeting, Jun 2018, Strasbourg, France. ⟨hal-03993195⟩
  • Lucile Brunel-Duverger, Sandrine Pagès-Camagna, Nancy Brodie-Linder, Hélène Guichard, Patricia Rigault-Déon, et al.. To the understanding of the complex manufacturing of Egyptian yellow coffins by non-invasive techniques. InArt, Mar 2018, Parma, Italy. ⟨hal-01715474⟩
  • Lucile Brunel-Duverger, Sandrine Pagès-Camagna, Nancy Brodie-Linder, Hélène Guichard, Anne Maigret, et al.. Pigment study of the 21st Egyptian Dynasty Yellow Coffins from the Louvre collection : analytical methodology and first results. Science of Ancient Egyptian Materials and Technologies Conference, Nov 2017, Cairo, Egypt. ⟨hal-01715427⟩
  • Lucile Brunel-Duverger, Sandrine Pagès-Camagna, Nancy Brodie-Linder, V Asensi Amoros, Juliette Langlois, et al.. Polychromy study of Yellow Coffins production, first results from Egyptian Antiquities Department objects . Second Vatican Coffin Conference, Musei Vaticani, Jun 2017, Vatican, Italy. ⟨hal-01715044⟩
  • Lucile Brunel-Duverger, Sandrine Pagès-Camagna. PILINA: investigating the use of precious hues on Greek figurines. Terres cuites Grecques et Romaines: 20 ans d'étude et de restauration, C2RMF et Musée du Louvre, Nov 2016, Paris, France. ⟨hal-01715032⟩
  • Lucie Vandromme, Li Chen, Lai Wei, Franck Le Bideau, André Loupy, et al.. Chiral imines on the wave: reactivity of tert-butyl acrylate and stereoselectivity determination using NMR in liquid crystals. MOL2NET, International Conference on Multidisciplinary Sciences, 2015, SCIForum, France. pp.1-18, ⟨10.3390/MOL2NET-1-a003⟩. ⟨hal-02314359⟩
  • Delphine Firley, Blandine Courcot, Jean-Michel Gillet, Anne Spasojevic - de Biré, Bernard Fraisse, et al.. Electrostatic properties of two precursors of potent HIV-1 integrase inhibitors. XX IUCR, Aug 2005, Florence, Italy. pp.c277 c277, ⟨10.1107/S0108767305088203⟩. ⟨hal-02304690⟩
  • M. Pizzonero, L. Keller, Françoise Dumas, M. Ourevitch, G. Morgant, et al.. Apports de la diffraction des rayons X et de la densité électronique expérimentale à l’étude d’intermédiaires de synthèse de la céphalotaxine. Rencontres de chimie organique Jeunes chercheurs, RCO 2004, SFC, Mar 2004, Versailles, France. ⟨hal-02304557⟩
  • M. Pizzonero, L. Keller, Françoise Dumas, M. Ourevitch, G. Morgant, et al.. Apports de la diffraction des rayons X et de la densité électronique expérimentale à l’étude d’intermédiaires de synthèse de la céphalotaxine. 11ème Journée Jeunes Chercheurs de la Société de Chimie Thérapeutique, Jan 2004, Paris, France. ⟨hal-02304554⟩
  • M. Pizzonero, L. Keller, Françoise Dumas, M. Ourevitch, G. Morgant, et al.. Charge density of a putative synthetic intermediate in the total synthesis of the cephalotaxine. Journées de la SFC-Champagne, Nov 2003, Reims, France. ⟨hal-02304551⟩
  • Goran A. Bogdanović, Anne Spasojevic - de Biré, Nour-Eddine Ghermani, M. Pizzonero, Françoise Dumas, et al.. Charge density of a putative intermediary product in the total synthesis of the cephalotaxine. XXI European Crystallographic Meeting, Aug 2003, Durban, South Africa. pp.24 - 29. ⟨hal-02304547⟩
  • Anne Spasojevic - de Biré, A. Kremenović, Nouhza Bouhmaida, G. Morgant, Nour-Eddine Ghermani. Experimental electron density of Zn-aspirinate complex: the subtlety of a 3d10 metal bonding to a drug-ligand. American Crystallographic Association Meeting, ACA-2002, May 2002, San Antonio, United States. ⟨hal-02304430⟩

Poster communications19 document

  • Marie Vayer. Mechanism-Guided Electrochemical N-Propargylation of N-Heterocycles via Decarboxylation of Allenoic Acids. JCO2025, Oct 2025, Palaiseau (Ecole Polytechnique), France. ⟨hal-05351029⟩
  • Nadège Lubin-Germain. Model-guided design of bactericidal agents from viral fusion peptides. ChemBioParis, Oct 2025, Paris, France. ⟨hal-05312268⟩
  • María Gutiérrez-Sánchez, H. Varet, P. Loiseau, S. Pomel, H. Lecoeur, et al.. Leishmania amazonensis exploits the macrophage epigenetic enzyme LSD1 for intracellular survival. EMBO Workshop - Host-parasite relationship: From mechanisms to control strategies, Oct 2025, Île des Embiez, 83140 Six-Fours-les-Plages, France. ⟨hal-05467152⟩
  • Marie Vayer. Mechanism-Guided Electrochemical N-Propargylation of N-Heterocycles via Decarboxylation of Allenoic Acids. OMCOS22, Sep 2025, Kyoto (Japan), Japan. ⟨hal-05351020⟩
  • Ines Carreira Costa, Margarida M Alves, Rita C. Guedes, José A. Paixão, Philippe M Loiseau, et al.. In silico and in vitro assessments of thio-linked pyrimidine-based compounds against Leishmania donovani. Congrès SFP SFMM, Jun 2025, Amiens, France. ⟨hal-05173348⟩
  • Camille Dejoux, Manuela Pastoriza-Gallego, Nadège Lubin-Germain, Simon Gonzalez, Abdelghani Oukhaled. Cell penetrating peptides probed by nanopores. Biophysical Society annual symposium, Feb 2025, Los Angeles, United States. . ⟨hal-05312263⟩
  • Linhua Shen, Olivier Monasson, Linhua Shen, Elisa Peroni, Franck Le Bideau, et al.. New electrochemical method for Arylation of Cysteine containing peptides. European Peptide symposium 2024, Aug 2024, Florence, Italy. ⟨hal-04724342⟩
  • Adrien Mourgout, F. Arjmand, E. Groult, Olivier Monasson, S. Ammar, et al.. Enhancing biomedical metal implants with synthetic peptides: improved bioactivity and in vitro safety. European Peptide symposium 2024, Aug 2024, Florence, Italy. ⟨hal-04727725⟩
  • Antoine Gamet, Ismaila Ciss, Bastien Nay. Total synthesis of photoactivatable latrunculin B for actin-targeting chemical biology. Rencontres de Chimie Organique, Apr 2024, Palaiseau (Université Paris-Saclay), France. ⟨hal-04575270⟩
  • Olivier Monasson, Alima Chali, Sonia Touharia, Adrien Mourgout, Farzin Arjmand, et al.. Novel biocompatible alloys via peptides surface engineering. A decade of Peptide Materials, Oct 2023, Sorrento, Italy. . ⟨hal-04725375⟩
  • David Rondeau, Thomas Delhaye, Erell Froger, Yves Gimbert, Axel Raux, et al.. Proposition of optimization strategies in collision energies on QTOF and Orbitrap instruments to perform comparable CID-MS-MS spectra in metabolomics. 39ème Journées Françaises de Spectrométrie de Masse (SFSM 2023 ), Sep 2023, Marseille, France. 2023. ⟨hal-04328759⟩
  • Enzo Lezin, Sarah Szwarc, Louis-Valentin Méteignier, Duchesse-Lacours Zamar, Caroline Birer Williams, et al.. The CYP71 Geissoschizine Cyclase catalyzes multiple cyclisation reactions in the synthesis of monoterpene indole alkaloids. P450 Biodiversity and Biotechnology, 2023, Copenhagen, Denmark. ⟨hal-05056241⟩
  • Enzo Lezin, Louis-Valentin Méteignier, Caroline Birer-Williams, Christelle Dutilleul, Arnaud Lanoue, et al.. Elucidating missing steps in the synthesis of the nootropic alkaloid vincamine and production of vincamine-derivatives by human P450s. 34eme colloque BioTechnoCentre, 2022, Nouan-le-Fuzelier, France. ⟨hal-05056191⟩
  • Louis-Valentin Méteignier, Caroline Birer Williams, Mehdi A. Beniddir, Pierre Le Pogam, Christelle Dutilleul, et al.. Transcriptomics in a tropical tree identify a P450 catalyzing distinct cyclizations of monoterpene indole alkaloids. 33eme colloque BioTechnoCentre, 2021, Chaumont sur Tharonne, France. ⟨hal-05055979⟩
  • T.M. Vishwanatha, D. Montoir, Mehdi Amoura, Z. El Ababsa, E. Yen-Pon, et al.. Synthesis of aryl-thioglycopeptides through chemoselective Pd-catalyzed conjugation. 26. American Peptide Symposium (APS 2019), Jun 2019, Monterey, Californie, United States. ⟨hal-02893419⟩
  • T.M. Vishwanatha, D. Montoir, Mehdi Amoura, Z. El Ababsa, E. Yen-Pon, et al.. Synthesis of aryl-thioglycopeptides through chemoselective Pd-catalyzed conjugation. 21. Réunion du Groupe Français des Peptides et des Protéines (GFPP21), May 2019, Amboise, France. ⟨hal-02893488⟩
  • David Montoir, Mehdi Amoura, Zine El Abidine Ababsa, Thimmalapura Marulappa Vishwanatha, Expédite Yen-Pon, et al.. Synthesis of aryl-Thioglycopeptides through chemoselective Pd-catalyzed conjugation. 35 th European Peptide Symposium, Aug 2018, Dublin, Ireland. 2018. ⟨hal-02734043⟩
  • Lucile Brunel-Duverger, V Asensi Amoros, Laurent Binet, Hélène Guichard, Elsa Lambert, et al.. AF 9590, a Yellow Coffin from the Egyptian Antiquities Department of the Louvre Museum: analytical methodology developped in the C2RMF within the Vatican Coffin Project . ICOM-CC, Sep 2017, Copenhagen, Denmark. 2017. ⟨hal-01715060⟩
  • Marion Alter, Anne-Solenn Le Hô, Myriam Eveno, Patrice Lehuédé, Sandrine Pages-Camagna, et al.. Conservation and alteration of painting pigments: the case of green copper-based organometallic pigments. Metal Soaps in Art, Mar 2016, Amsterdam, Netherlands. ⟨hal-01289465⟩

Proceedings1 document

  • Lorenzo Meneghelli, Lamia El Guermah, Maud Larregola, Sabrina Kellouche-Gaillard, Franck Carreiras, et al.. Design and Synthesis of Pin1-PROTACs as Potential Therapeutic Tools for Cancer Treatment. 36th European Peptide Symposium, Aug 2022, Sitges (Barcelona), Spain. The European Peptide Society, pp.285-287, 2022, ⟨10.17952/36EPS/36EPS.2022.285⟩. ⟨hal-05003974⟩

Book sections12 document

  • Pierre Milbéo, Chiara Zanato. The Thiol-ene “Click” Reaction for Synthesis of Biomolecular Thioether and Thioester Derivatives. Topics Heterocyclic Chemistry. Modern Advances in Click Chemistry: Synthesis of Compounds, Springer Berlin Heidelberg, In press, Topics in Heterocyclic Chemistry, ⟨10.1007/7081_2025_98⟩. ⟨hal-05479896⟩
  • A Ferry, Florian Gallier, S Gonzalez, N Lubin-Germain, L Soter de Mariz E Miranda, et al.. Enabling technologies applied to glycosylation. Carbohydrate Chemistry: Chemical and Biological Approaches, 46, pp.44-72, 2024, 978-1-83767-217-2. ⟨10.1039/9781837672844-00044⟩. ⟨hal-05352935⟩
  • Thierry Brigaud, B. Crousse, T. Lequeux. Perfluoroalkylated Biomolecules for Medicinal Chemistry and Biological Studies. Perfluoroalkyl Substances, The Royal Society of Chemistry; The Royal Society of Chemistry, pp.459-476, 2022, ⟨10.1039/9781839167591-00459⟩. ⟨hal-04098116⟩
  • Pierre Le Pogam, Erwan Poupon, Pierre Champy, Mehdi Beniddir. Implementation of an MS/MS Spectral Library for Monoterpene Indole Alkaloids. Catharanthus roseus, 2505, Springer US, pp.87-100, 2022, Methods in Molecular Biology, ⟨10.1007/978-1-0716-2349-7_7⟩. ⟨hal-05058417⟩
  • Angélique Ferry, Xavier Guinchard. Bicyclic 5-5 Systems With One Bridgehead (Ring Junction) Nitrogen Atom: Two Extra Heteroatoms 1:1. Comprehensive Heterocyclic Chemistry IV, Elsevier, pp.95-144, 2022, ⟨10.1016/B978-0-12-409547-2.14934-0⟩. ⟨hal-04102152⟩
  • Angélique Ferry, Florian Gallier, Simon Gonzalez, Nadège Lubin-Germain, Leandro Soter de Mariz E Miranda, et al.. Recent advances in the functionalization of unprotected carbohydrates. Amélia Pilar Rauter; Thisbe K Lindhorst; Yves Queneau. Carbohydrate Chemistry: Chemical and Biological Approaches, 45, Royal Society of Chemistry, pp.239-304, 2021, SPR - Carbohydrate Chemistry, 978-1-83916-390-6. ⟨10.1039/9781839164538-00239⟩. ⟨hal-03667486⟩
  • Laurent Ferrié. Advances in the synthesis of 1,2-dioxolanes and 1,2-dioxanes. Eric F.V. Scriven; Christopher A. Ramsden. Advances in Heterocyclic Chemistry, 135, Elsevier, pp.57-146, 2021, 978-0-12-824619-1. ⟨10.1016/bs.aihch.2021.03.001⟩. ⟨hal-03320615⟩
  • Benoit Crousse, Thierry Milcent. Synthesis of NCF3, NCF2H and NCH2CF3 motifs. merging Fluorinated Motifs. Properties, Synthesis and Applications, 2020. ⟨hal-03796648⟩
  • Mouad Alami. De nouvelles perspectives en thérapie antivasculaire Pourquoi faire compliquer quand on peut faire simple ?. Chimie et biologie de synthèse. Les applications, 2019, ⟨10.1051/978-2-7598-2316-1.c017⟩. ⟨hal-02414134⟩
  • Chantal Andraud, Philippe Belmont, J.M. Campagne, Gaëlle Chouraqui, Emmanuel Gras, et al.. Rapport de Conjoncture du CoNRS 2014 (INC / Section 12). CNRS Editions, Paris,. Rapport de Conjoncture du CoNRS 2014, CNRS Editions, Paris,, pp.255-274, 2014, 978-2-271-08746-1. ⟨hal-02338362⟩
  • Danièle Bonnet-Delpon, Jean-Pierre Bégué, Benoit Crousse, Fabienne Grellepois, Constance Chollet, et al.. New 10-Trifluoromethyl Monomers, Dimers, and Chimeras of Artemisinin from a Key Allyl Bromide Precursor. Current fluoroorganic chemistry: new synthetic directions, technologies, materials and biological application, ACS Symposium Series, Vol 949, pp.337-351, 2007, ⟨10.1021/bk-2007-0949.ch020⟩. ⟨mnhn-02867458⟩
  • Jean-Hugues Renault, Jean-Marc Nuzillard, Olivier Intes, Alexandre Maciuk. Solvent systems. Alain Berthod. Comprehensive Analytical Chemistry Series, 38, Elsevier, pp.49-83, 2005, Countercurrent chromatography, the support-free liquid stationary phase, 978-0444507372. ⟨10.1016/S0166-526X(02)80006-X⟩. ⟨hal-01968195⟩

Patents1 document

  • Maité Sylla-Iyarreta Veitía, Françoise Dumas, Georges Morgant. Synthesis Characterization and biological activities of metal-base complexes containing the leading drug valproic acid. France, Patent n° : PCT/FR2009/051077. 2009. ⟨hal-01487516⟩

Preprints, Working Papers13 document

  • Mohammed Latrache, Amina Sesay, Samuel Oger, Mireia Benito Montaner, Jinlei Zhang, et al.. Bioinspired Synthesis of Sceptrin, Ageliferin and Six Piperine Dimers by Photo(Flow) catalysis: [2+2] vs [4+2] Cycloaddition. 2025. ⟨hal-05237335⟩
  • Flavio Alvarez, Florence Larrous, Ariel Mechaly, Benjamin Bardiaux, Quentin Goor, et al.. HTRF-based identification of small molecules targeting SARS-CoV-2 E protein interaction with ZO-1 PDZ2. 2025. ⟨pasteur-05261353⟩
  • Sandrine Ongeri, Benoît Crousse. Fluorinated triazolamers: preferential conformations and activities on Islet Amyloid Polypeptide (hIAPP) Aggregation. 2025. ⟨hal-05179626⟩
  • Yassine Mejri, Olivier Cailloux, Elvis Otogo N'Nang, Blandine Séon-Méniel, Jean-François Gallard, et al.. MS2DECIDE: Aggregating Multi-Annotated Tandem Mass Spectrometry Data with Decision Theory Enhances Natural Products Prioritization. 2025. ⟨hal-05058403⟩
  • Davide Di Lorenzo, Nicolo Bisi, Julia Kaffy, Lisa Marie Ramirez, Markus Zweckstetter, et al.. Synthetic chaperone based on Hsp90-Tau interaction inhibits pathological Tau aggregation and rescues physiological Tau-Microtubule interaction. 2025. ⟨hal-05047264⟩
  • Laurent Ferrié, Bruno Figadère, Nicolas Jamey, Bastien Champciaux. Peroxy-Carbenium Mediated Asymmetric Synthesis of 1,2-Dioxanes and 1,2-Dioxolanes. 2024. ⟨hal-04757792⟩
  • Florent Dumont, Emy Ponsardin, Guillaume Bernadat, Sylvia Cohen-Kaminsky. MOAL: Multi-Omic Analysis at Lab. A simplified methodology workflow to make reproducible omic bioanalysis. 2023. ⟨hal-04294241⟩
  • José Laxio Arenas, Jacopo Lesma, Tap Ha-Duong, Bikash Sahoo, Ayyalusamy Ramamoorthy, et al.. Relation between conformation and activity on islet amyloid polypeptide aggregation of fluorinated foldamers based on Ndifluoromethyl-1,4-triazole amino acids. 2023. ⟨hal-04273096⟩
  • Yazid Boutahri, Khoubaib Ben Haj Salah, Nicolas Tisserand, Nathalie Lensen, Benoit Crousse, et al.. Difluoroalanine: Synthesis, Incorporation in Peptides, and Hydrophobic Contribution Assessment. 2023. ⟨hal-04249424⟩
  • Clémence Rose, Rodrigo Hernán Tomas-Grau, Brenda Zabala, Jean-Michel Brunel, Patrick Michel, et al.. Enhancing Inhibition of Both α-Synuclein Aggregation and Neuroinflammation: New Insights into the C-9 Modification of Doxycycline. 2023. ⟨hal-04250582⟩
  • Mansour Dolé Kérim, Laurent Evanno, Laurent Ferrie. Stereodivergent Total Syntheses of (+)-Mycaperoxides C, D, G Methyl Ester and (-)-Mycaperoxide B. 2022. ⟨hal-03775643⟩
  • Marion Barthé, Flora Lefebvre, Emilie Langlois, Florence Lefebvre, Patrick Lechêne, et al.. PEGylated isoprenaline reveals distinct functions of cardiac β-adrenergic receptors located in the T-tubule vs . outer surface membrane. 2022. ⟨hal-03793970⟩
  • Damien Olivier-Jimenez, Zakaria Bouchouireb, Simon Ollivier, Julia Mocquard, Pierre-Marie Allard, et al.. From mass spectral features to molecules in molecular networks : a novel workflow for untargeted metabolomics. 2021. ⟨hal-05098952⟩

Reports1 document

  • Fabrice Nesslany, Sabrina Boutefnouchet, Pierre Champy, Hanh Dufat, Marion Girardot, et al.. Avis de l'Anses relatif à l’évaluation des effets indésirables liés à la consommation de compléments alimentaires contenant du « Garcinia cambogia ». Saisine n°2020-SA-0047, Anses. 2025, 69 p. ⟨anses-05175504⟩

Theses31 document

  • Linlin Li. New approaches to the synthesis of S-and N-glycosides and C-furanosides. Organic chemistry. Université Paris-Saclay, 2025. English. ⟨NNT : 2025UPASQ048⟩. ⟨tel-05426219⟩
  • Sarah Szwarc. Développements méthodologiques en chimie analytique pour l'identification des enzymes catalysant des cyclisations C-N chez les alcaloïdes indolomonoterpéniques. Chimie analytique. Université Paris-Saclay, 2024. Français. ⟨NNT : 2024UPASQ074⟩. ⟨tel-05075853⟩
  • Sarah Szwarc. Développements méthodologiques en chimie analytique pour l'identification des enzymes catalysant des cyclisations C-N chez les alcaloïdes indolomonoterpéniques. Chimie analytique. Université Paris-Saclay, 2024. Français. ⟨NNT : 2024UPASQ074⟩. ⟨tel-05106245⟩
  • Vanessa Mussard. Conception d'une nouvelle classe de sondes photoisomérisables fluorescentes “off-on” pour l'étude de l'allostérie des protéines. Chimie organique. Université Paris-Saclay, 2024. Français. ⟨NNT : 2024UPASQ014⟩. ⟨tel-05396328⟩
  • María Gutiérrez Sánchez. Macrophage Lysine Demethylase LSD1 : Implications for intracellular Leishmania survival and host-directed drug discovery.. Cell Behavior [q-bio.CB]. Université Paris-Saclay, 2023. English. ⟨NNT : 2023UPASQ042⟩. ⟨tel-04290331⟩
  • Kaliroi Peqini. Development of molecular probes acting on Tau/Tubulin and a-Synuclein/Tubulin interface. Medicinal Chemistry. Université Paris-Saclay; Università degli studi (Milan, Italie). Dipartimento di Scienze della Terra, 2023. English. ⟨NNT : 2023UPASQ036⟩. ⟨tel-04662379⟩
  • Davide Di Lorenzo. Using β-strand and β-hairpin peptidomimetics induced by constrained amino acids to modulate the aggregation of the microtubule associated protein Tau : design, synthesis and evaluation. Medicinal Chemistry. Université Paris-Saclay; Università degli studi (Milan, Italie). Convegno di studi (2000 ; Milano), 2023. English. ⟨NNT : 2023UPASQ032⟩. ⟨tel-05215017⟩
  • Mayssa Zayene. Conception, synthèse et valorisation biologique de nouveaux dérivés tropines et tropanes. Chimie organique. Université Paris-Saclay; Université de Monastir (Tunisie), 2023. Français. ⟨NNT : 2023UPASQ028⟩. ⟨tel-04639064⟩
  • Phuong Y Mai. Exploration ciblée de l'espace chimique des micro-organismes des « mares de kopara » polynésiennes. Chimie analytique. Université Paris-Saclay, 2023. Français. ⟨NNT : 2023UPASQ003⟩. ⟨tel-04536647⟩
  • Tingting Cao. Design and synthesis of new fluorinated hydrazines. Organic chemistry. Université Paris-Saclay, 2022. English. ⟨NNT : 2022UPASQ072⟩. ⟨tel-04058237⟩
  • Maxence Delaunay. Conception in silico d'inhibiteurs peptidiques d'interactions protéine-protéine. Bio-Informatique, Biologie Systémique [q-bio.QM]. Université Paris-Saclay, 2022. Français. ⟨NNT : 2022UPASQ069⟩. ⟨tel-04022527⟩
  • Zineb Fechtali Moute. Etude de la biodiversité et de la viabilité des amibes libres dans un réseau d'eau potable : approches environnementales et fondamentales. Parasitologie. Université Paris-Saclay, 2022. Français. ⟨NNT : 2022UPASQ062⟩. ⟨tel-04672721⟩
  • Chenghui Shi. Synthesis and conformational analysis of peptidomimetic foldamers containing diaza-peptide units : application in protein-protein interactions. Molecular biology. Université Paris-Saclay, 2022. English. ⟨NNT : 2022UPASQ055⟩. ⟨tel-04815486⟩
  • Ismaila Ciss. Synthèse totale des amphidinolides C et U. Chimie organique. Université Paris-Saclay; Université Cheikh Anta Diop (Dakar, Sénégal ; 1957-..), 2022. Français. ⟨NNT : 2022UPASQ039⟩. ⟨tel-04215937⟩
  • Mingxiang Zhu. New approaches to the synthesis of S/Se-glycosides and alkynyl C-nucleosides. Catalysis. Université Paris-Saclay, 2022. English. ⟨NNT : 2022UPASQ030⟩. ⟨tel-04153055⟩
  • Nedjwa Bennai. Étude de la réactivité des sucres dans les couplages organométalliques : application à la synthèse de glycosides biologiquement actifs. Chimie organique. Université Paris-Saclay; Université des Sciences et de la Technologie d'Oran Mohamed-Boudiaf (Algérie), 2022. Français. ⟨NNT : 2022UPASQ016⟩. ⟨tel-03681327⟩
  • Elodie Pradayrol. Vers la synthèse biomimétique de pigments fongiques : la sclérocitrine et la chalcitrine. Etude des métabolites de Scleroderma citrinum. Chimie organique. Université Paris-Saclay, 2022. Français. ⟨NNT : 2022UPASQ005⟩. ⟨tel-03662479⟩
  • José Laxio Arenas. Triazolamères fluorés : conception, synthèse, études conformationnelles et modulation de l'agrégation de peptides amyloïdes. Chimie thérapeutique. Université Paris-Saclay, 2022. Français. ⟨NNT : 2022UPASQ003⟩. ⟨tel-03962087⟩
  • Juba Ghouilem. Une nouvelle approche d'activation C(sp³) -H de sucres : vers de nouvelles classes de glycomimétiques C-hétérosides. Chimie organique. Université Paris-Saclay, 2021. Français. ⟨NNT : 2021UPASQ053⟩. ⟨tel-04334442⟩
  • Aminata Ouayogode. Etude ethnobotanique, chimique et activités pharmacologiques de plantes et recettes antimalariques de Côte d’Ivoire. Chimie thérapeutique. Université Paris-Saclay; Université Félix Houphouët-Boigny (Abidjan, Côte d'Ivoire), 2021. Français. ⟨NNT : 2021UPASQ034⟩. ⟨tel-03650772⟩
  • Sen Wang. Synthèse et fonctionnalisation d'azobenzènes : vers le développement de sondes photocommutables. Chimie organique. Université Paris-Saclay, 2021. Français. ⟨NNT : 2021UPASQ013⟩. ⟨tel-03341233⟩
  • Victor Turpin. Hypothèses de biosynthèse des alcaloïdes indolomonoterpéniques : résolution de mécanismes fondamentaux par la synthèse et par la modélisation. Chimie organique. Université Paris-Saclay, 2021. Français. ⟨NNT : 2021UPASQ009⟩. ⟨tel-03578052⟩
  • Jacopo Lesma. β-Hairpin peptidomimetics as inhibitors of hIAPP amyloid protein aggregation : design, synthesis and evaluation. Medicinal Chemistry. Université Paris-Saclay, 2020. English. ⟨NNT : 2020UPASQ018⟩. ⟨tel-03793799⟩
  • Charlotte Alcover. Réseaux moléculaires et Chimie des Substances Naturelles : de l’isolement de composés inédits à de toutes nouvelles applications en synthèse biomimétique. Chimie organique. Université Paris Saclay (COmUE), 2019. Français. ⟨NNT : 2019SACLS569⟩. ⟨tel-03506234⟩
  • Maud Chan Yao Chong. Structure et dynamique de protéines intrinsèquement désordonnées : Caractérisation par une approche combinant dynamique moléculaire avancée et SAXS. Biologie structurale [q-bio.BM]. Université Paris Saclay (COmUE), 2019. Français. ⟨NNT : 2019SACLS257⟩. ⟨tel-02968589⟩
  • Oussema Ouerfelli. Aziridine-2-carboxylates et leurs dérivées : Nouvelles perspectives en synthèse hétérocycliques et chimie des peptides.. Chimie analytique. Université de Cergy Pontoise; Université de Tunis El Manar, 2018. Français. ⟨NNT : 2018CERG0973⟩. ⟨tel-02285887⟩
  • Siguara Bastos de Lemos E Silva. Chemistry and biosynthesis of highly complex marine alkaloids from Mediterranean biodiversity. Organic chemistry. Université Paris Saclay (COmUE), 2017. English. ⟨NNT : 2017SACLS214⟩. ⟨tel-02953258⟩
  • Matthaia Ieronymaki. Immunological and Conformational characterization of synthetic peptide probes for autoimmune diseases. Human health and pathology. Université de Cergy Pontoise, 2016. English. ⟨NNT : 2016CERG0831⟩. ⟨tel-01470760⟩
  • Elodie Jagu. Design, synthesis and biological evaluation of new polyamine derivatives as antikinetoplastid agents. Organic chemistry. Université Paris Saclay (COmUE), 2016. English. ⟨NNT : 2016SACLS589⟩. ⟨tel-01654426⟩
  • Nicolo Tonali. Synthetic mimics of beta-sheets : design, synthesis and evaluation of their ability to modulate the aggregation of the beta-amyloid 1-42 peptide.. Medicinal Chemistry. Université Paris-Saclay, 2016. English. ⟨NNT : 2016SACLS544⟩. ⟨tel-01933728⟩
  • Cédric Rentier. Autoimmune diseases : design, synthesis and immunological screening of post-translationally modified peptides to characterize autoantibodies in patients' sera. Organic chemistry. Université de Cergy Pontoise; Università degli Studi di Firenze, 2015. English. ⟨NNT : 2015CERG0746⟩. ⟨tel-01214960⟩

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